DrugRepV Browse Page


DrugRepV browse page allows user to take a glance of the particular antiviral agent.Fields in the webpage is hylerlinked ot various external repositories like DrugBank, PubChem, Clinicaltrials.gov,and PubMed.User can explore the biological, Clinical, Chemical, and Structural details of every repurposed drug candidate.By clicking on the table header arrows, user can sort entries in ascending or descending order.


Total number of Records for Single-round viral replication assay are 290




DrugRepV_ID Antiviral Name
Drug type
Primary Indication
Secondary Indication
Strain
Pathways
Assay
Activity
Clinical Status
References
DrugRepV_6577Raltegravir
Antiinfectives For Systemic Use
Acquired immunodeficiency syndrome
Human immunodeficiency virus
WT
Pathway
Single-round viral replication assay
Decrease (50 %)
Approved
29769116
DrugRepV_6578Raltegravir
Antiinfectives For Systemic Use
Acquired immunodeficiency syndrome
Human immunodeficiency virus
Y143R (RAL)
Pathway
Single-round viral replication assay
Decrease (50 %)
Approved
29769116
DrugRepV_6579Raltegravir
Antiinfectives For Systemic Use
Acquired immunodeficiency syndrome
Human immunodeficiency virus
N155H(RAL)
Pathway
Single-round viral replication assay
Decrease (50 %)
Approved
29769116
DrugRepV_6580Raltegravir
Antiinfectives For Systemic Use
Acquired immunodeficiency syndrome
Human immunodeficiency virus
G140S/Q148H (RAL)
Pathway
Single-round viral replication assay
Decrease (50 %)
Approved
29769116
DrugRepV_6581Raltegravir
Antiinfectives For Systemic Use
Acquired immunodeficiency syndrome
Human immunodeficiency virus
T661(EVG)
Pathway
Single-round viral replication assay
Decrease (50 %)
Approved
29769116
DrugRepV_6582Raltegravir
Antiinfectives For Systemic Use
Acquired immunodeficiency syndrome
Human immunodeficiency virus
E92Q (EVG)
Pathway
Single-round viral replication assay
Decrease (50 %)
Approved
29769116
DrugRepV_6583Raltegravir
Antiinfectives For Systemic Use
Acquired immunodeficiency syndrome
Human immunodeficiency virus
H51Y (DTG)
Pathway
Single-round viral replication assay
Decrease (50 %)
Approved
29769116
DrugRepV_6584Raltegravir
Antiinfectives For Systemic Use
Acquired immunodeficiency syndrome
Human immunodeficiency virus
G118R (DTG)
Pathway
Single-round viral replication assay
Decrease (50 %)
Approved
29769116
DrugRepV_6585Raltegravir
Antiinfectives For Systemic Use
Acquired immunodeficiency syndrome
Human immunodeficiency virus
R263K (DTG)
Pathway
Single-round viral replication assay
Decrease (50 %)
Approved
29769116
DrugRepV_6586Raltegravir
Antiinfectives For Systemic Use
Acquired immunodeficiency syndrome
Human immunodeficiency virus
H51Y/R263K (DTG)
Pathway
Single-round viral replication assay
Decrease (50 %)
Approved
29769116
DrugRepV_6587Raltegravir
Antiinfectives For Systemic Use
Acquired immunodeficiency syndrome
Human immunodeficiency virus
E138K/R263K (DTG)
Pathway
Single-round viral replication assay
Decrease (50 %)
Approved
29769116
DrugRepV_6588Elvitegravir
Antiinfectives For Systemic Use
Acquired immunodeficiency syndrome
Human immunodeficiency virus
WT
Pathway
Single-round viral replication assay
Decrease (50 %)
Approved
29769116
DrugRepV_6589Elvitegravir
Antiinfectives For Systemic Use
Acquired immunodeficiency syndrome
Human immunodeficiency virus
Y143R (RAL)
Pathway
Single-round viral replication assay
Decrease (50 %)
Approved
29769116
DrugRepV_6590Elvitegravir
Antiinfectives For Systemic Use
Acquired immunodeficiency syndrome
Human immunodeficiency virus
N155H(RAL)
Pathway
Single-round viral replication assay
Decrease (50 %)
Approved
29769116
DrugRepV_6591Elvitegravir
Antiinfectives For Systemic Use
Acquired immunodeficiency syndrome
Human immunodeficiency virus
G140S/Q148H (RAL)
Pathway
Single-round viral replication assay
Decrease (50 %)
Approved
29769116
DrugRepV_6592Elvitegravir
Antiinfectives For Systemic Use
Acquired immunodeficiency syndrome
Human immunodeficiency virus
T661(EVG)
Pathway
Single-round viral replication assay
Decrease (50 %)
Approved
29769116
DrugRepV_6593Elvitegravir
Antiinfectives For Systemic Use
Acquired immunodeficiency syndrome
Human immunodeficiency virus
E92Q (EVG)
Pathway
Single-round viral replication assay
Decrease (50 %)
Approved
29769116
DrugRepV_6594Elvitegravir
Antiinfectives For Systemic Use
Acquired immunodeficiency syndrome
Human immunodeficiency virus
H51Y (DTG)
Pathway
Single-round viral replication assay
Decrease (50 %)
Approved
29769116
DrugRepV_6595Elvitegravir
Antiinfectives For Systemic Use
Acquired immunodeficiency syndrome
Human immunodeficiency virus
G118R (DTG)
Pathway
Single-round viral replication assay
Decrease (50 %)
Approved
29769116
DrugRepV_6596Elvitegravir
Antiinfectives For Systemic Use
Acquired immunodeficiency syndrome
Human immunodeficiency virus
R263K (DTG)
Pathway
Single-round viral replication assay
Decrease (50 %)
Approved
29769116
DrugRepV_6597Elvitegravir
Antiinfectives For Systemic Use
Acquired immunodeficiency syndrome
Human immunodeficiency virus
H51Y/R263K (DTG)
Pathway
Single-round viral replication assay
Decrease (50 %)
Approved
29769116
DrugRepV_6598Elvitegravir
Antiinfectives For Systemic Use
Acquired immunodeficiency syndrome
Human immunodeficiency virus
E138K/R263K (DTG)
Pathway
Single-round viral replication assay
Decrease (50 %)
Approved
29769116
DrugRepV_6599Dolutegravir
Antiinfectives For Systemic Use
Acquired immunodeficiency syndrome
Human immunodeficiency virus
WT
Pathway
Single-round viral replication assay
Decrease (50 %)
Approved
29769116
DrugRepV_6600Dolutegravir
Antiinfectives For Systemic Use
Acquired immunodeficiency syndrome
Human immunodeficiency virus
Y143R (RAL)
Pathway
Single-round viral replication assay
Decrease (50 %)
Approved
29769116
DrugRepV_6601Dolutegravir
Antiinfectives For Systemic Use
Acquired immunodeficiency syndrome
Human immunodeficiency virus
N155H(RAL)
Pathway
Single-round viral replication assay
Decrease (50 %)
Approved
29769116
DrugRepV_6602Dolutegravir
Antiinfectives For Systemic Use
Acquired immunodeficiency syndrome
Human immunodeficiency virus
G140S/Q148H (RAL)
Pathway
Single-round viral replication assay
Decrease (50 %)
Approved
29769116
DrugRepV_6603Dolutegravir
Antiinfectives For Systemic Use
Acquired immunodeficiency syndrome
Human immunodeficiency virus
T661(EVG)
Pathway
Single-round viral replication assay
Decrease (50 %)
Approved
29769116
DrugRepV_6604Dolutegravir
Antiinfectives For Systemic Use
Acquired immunodeficiency syndrome
Human immunodeficiency virus
E92Q (EVG)
Pathway
Single-round viral replication assay
Decrease (50 %)
Approved
29769116
DrugRepV_6605Dolutegravir
Antiinfectives For Systemic Use
Acquired immunodeficiency syndrome
Human immunodeficiency virus
H51Y (DTG)
Pathway
Single-round viral replication assay
Decrease (50 %)
Approved
29769116
DrugRepV_6606Dolutegravir
Antiinfectives For Systemic Use
Acquired immunodeficiency syndrome
Human immunodeficiency virus
G118R (DTG)
Pathway
Single-round viral replication assay
Decrease (50 %)
Approved
29769116
DrugRepV_6607Dolutegravir
Antiinfectives For Systemic Use
Acquired immunodeficiency syndrome
Human immunodeficiency virus
R263K (DTG)
Pathway
Single-round viral replication assay
Decrease (50 %)
Approved
29769116
DrugRepV_6608Dolutegravir
Antiinfectives For Systemic Use
Acquired immunodeficiency syndrome
Human immunodeficiency virus
H51Y/R263K (DTG)
Pathway
Single-round viral replication assay
Decrease (50 %)
Approved
29769116
DrugRepV_6609Dolutegravir
Antiinfectives For Systemic Use
Acquired immunodeficiency syndrome
Human immunodeficiency virus
E138K/R263K (DTG)
Pathway
Single-round viral replication assay
Decrease (50 %)
Approved
29769116
DrugRepV_6610Cabotegravir
Antiviral
Acquired immunodeficiency syndrome
Human immunodeficiency virus
WT
Pathway
Single-round viral replication assay
Decrease (50 %)
Phase I
29769116
DrugRepV_6611Cabotegravir
Antiviral
Acquired immunodeficiency syndrome
Human immunodeficiency virus
Y143R (RAL)
Pathway
Single-round viral replication assay
Decrease (50 %)
Phase I
29769116
DrugRepV_6612Cabotegravir
Antiviral
Acquired immunodeficiency syndrome
Human immunodeficiency virus
N155H(RAL)
Pathway
Single-round viral replication assay
Decrease (50 %)
Phase I
29769116
DrugRepV_6613Cabotegravir
Antiviral
Acquired immunodeficiency syndrome
Human immunodeficiency virus
G140S/Q148H (RAL)
Pathway
Single-round viral replication assay
Decrease (50 %)
Phase I
29769116
DrugRepV_6614Cabotegravir
Antiviral
Acquired immunodeficiency syndrome
Human immunodeficiency virus
T661(EVG)
Pathway
Single-round viral replication assay
Decrease (50 %)
Phase I
29769116
DrugRepV_6615Cabotegravir
Antiviral
Acquired immunodeficiency syndrome
Human immunodeficiency virus
E92Q (EVG)
Pathway
Single-round viral replication assay
Decrease (50 %)
Phase I
29769116
DrugRepV_6616Cabotegravir
Antiviral
Acquired immunodeficiency syndrome
Human immunodeficiency virus
H51Y (DTG)
Pathway
Single-round viral replication assay
Decrease (50 %)
Phase I
29769116
DrugRepV_6617Cabotegravir
Antiviral
Acquired immunodeficiency syndrome
Human immunodeficiency virus
G118R (DTG)
Pathway
Single-round viral replication assay
Decrease (50 %)
Phase I
29769116
DrugRepV_6618Cabotegravir
Antiviral
Acquired immunodeficiency syndrome
Human immunodeficiency virus
R263K (DTG)
Pathway
Single-round viral replication assay
Decrease (50 %)
Phase I
29769116
DrugRepV_6619Cabotegravir
Antiviral
Acquired immunodeficiency syndrome
Human immunodeficiency virus
H51Y/R263K (DTG)
Pathway
Single-round viral replication assay
Decrease (50 %)
Phase I
29769116
DrugRepV_6620Cabotegravir
Antiviral
Acquired immunodeficiency syndrome
Human immunodeficiency virus
E138K/R263K (DTG)
Pathway
Single-round viral replication assay
Decrease (50 %)
Phase I
29769116
DrugRepV_6621Bictegravir
Antiinfectives For Systemic Use
Acquired immunodeficiency syndrome
Human immunodeficiency virus
WT
Pathway
Single-round viral replication assay
Decrease (50 %)
Approved
29769116
DrugRepV_6622Bictegravir
Antiinfectives For Systemic Use
Acquired immunodeficiency syndrome
Human immunodeficiency virus
Y143R (RAL)
Pathway
Single-round viral replication assay
Decrease (50 %)
Approved
29769116
DrugRepV_6623Bictegravir
Antiinfectives For Systemic Use
Acquired immunodeficiency syndrome
Human immunodeficiency virus
N155H(RAL)
Pathway
Single-round viral replication assay
Decrease (50 %)
Approved
29769116
DrugRepV_6624Bictegravir
Antiinfectives For Systemic Use
Acquired immunodeficiency syndrome
Human immunodeficiency virus
G140S/Q148H (RAL)
Pathway
Single-round viral replication assay
Decrease (50 %)
Approved
29769116
DrugRepV_6625Bictegravir
Antiinfectives For Systemic Use
Acquired immunodeficiency syndrome
Human immunodeficiency virus
T661(EVG)
Pathway
Single-round viral replication assay
Decrease (50 %)
Approved
29769116
DrugRepV_6626Bictegravir
Antiinfectives For Systemic Use
Acquired immunodeficiency syndrome
Human immunodeficiency virus
E92Q (EVG)
Pathway
Single-round viral replication assay
Decrease (50 %)
Approved
29769116
DrugRepV_6627Bictegravir
Antiinfectives For Systemic Use
Acquired immunodeficiency syndrome
Human immunodeficiency virus
H51Y (DTG)
Pathway
Single-round viral replication assay
Decrease (50 %)
Approved
29769116
DrugRepV_6628Bictegravir
Antiinfectives For Systemic Use
Acquired immunodeficiency syndrome
Human immunodeficiency virus
G118R (DTG)
Pathway
Single-round viral replication assay
Decrease (50 %)
Approved
29769116
DrugRepV_6629Bictegravir
Antiinfectives For Systemic Use
Acquired immunodeficiency syndrome
Human immunodeficiency virus
R263K (DTG)
Pathway
Single-round viral replication assay
Decrease (50 %)
Approved
29769116
DrugRepV_6630Bictegravir
Antiinfectives For Systemic Use
Acquired immunodeficiency syndrome
Human immunodeficiency virus
H51Y/R263K (DTG)
Pathway
Single-round viral replication assay
Decrease (50 %)
Approved
29769116
DrugRepV_6631Bictegravir
Antiinfectives For Systemic Use
Acquired immunodeficiency syndrome
Human immunodeficiency virus
E138K/R263K (DTG)
Pathway
Single-round viral replication assay
Decrease (50 %)
Approved
29769116
DrugRepV_6632Raltegravir
Antiinfectives For Systemic Use
Acquired immunodeficiency syndrome
Human immunodeficiency virus
M50I
Pathway
Single-round viral replication assay
Decrease (50 %)
Approved
29769116
DrugRepV_6633Raltegravir
Antiinfectives For Systemic Use
Acquired immunodeficiency syndrome
Human immunodeficiency virus
L74M
Pathway
Single-round viral replication assay
Decrease (50 %)
Approved
29769116
DrugRepV_6634Raltegravir
Antiinfectives For Systemic Use
Acquired immunodeficiency syndrome
Human immunodeficiency virus
T97A
Pathway
Single-round viral replication assay
Decrease (50 %)
Approved
29769116
DrugRepV_6635Raltegravir
Antiinfectives For Systemic Use
Acquired immunodeficiency syndrome
Human immunodeficiency virus
S119R
Pathway
Single-round viral replication assay
Decrease (50 %)
Approved
29769116
DrugRepV_6636Raltegravir
Antiinfectives For Systemic Use
Acquired immunodeficiency syndrome
Human immunodeficiency virus
E138K
Pathway
Single-round viral replication assay
Decrease (50 %)
Approved
29769116
DrugRepV_6637Raltegravir
Antiinfectives For Systemic Use
Acquired immunodeficiency syndrome
Human immunodeficiency virus
G140S
Pathway
Single-round viral replication assay
Decrease (50 %)
Approved
29769116
DrugRepV_6638Raltegravir
Antiinfectives For Systemic Use
Acquired immunodeficiency syndrome
Human immunodeficiency virus
Q146L
Pathway
Single-round viral replication assay
Decrease (50 %)
Approved
29769116
DrugRepV_6639Raltegravir
Antiinfectives For Systemic Use
Acquired immunodeficiency syndrome
Human immunodeficiency virus
Q146P
Pathway
Single-round viral replication assay
Decrease (50 %)
Approved
29769116
DrugRepV_6640Raltegravir
Antiinfectives For Systemic Use
Acquired immunodeficiency syndrome
Human immunodeficiency virus
Q148H
Pathway
Single-round viral replication assay
Decrease (50 %)
Approved
29769116
DrugRepV_6641Raltegravir
Antiinfectives For Systemic Use
Acquired immunodeficiency syndrome
Human immunodeficiency virus
Q148K
Pathway
Single-round viral replication assay
Decrease (50 %)
Approved
29769116
DrugRepV_6642Raltegravir
Antiinfectives For Systemic Use
Acquired immunodeficiency syndrome
Human immunodeficiency virus
Q148R
Pathway
Single-round viral replication assay
Decrease (50 %)
Approved
29769116
DrugRepV_6643Raltegravir
Antiinfectives For Systemic Use
Acquired immunodeficiency syndrome
Human immunodeficiency virus
S153Y
Pathway
Single-round viral replication assay
Decrease (50 %)
Approved
29769116
DrugRepV_6644Elvitegravir
Antiinfectives For Systemic Use
Acquired immunodeficiency syndrome
Human immunodeficiency virus
M50I
Pathway
Single-round viral replication assay
Decrease (50 %)
Approved
29769116
DrugRepV_6645Elvitegravir
Antiinfectives For Systemic Use
Acquired immunodeficiency syndrome
Human immunodeficiency virus
L74M
Pathway
Single-round viral replication assay
Decrease (50 %)
Approved
29769116
DrugRepV_6646Elvitegravir
Antiinfectives For Systemic Use
Acquired immunodeficiency syndrome
Human immunodeficiency virus
T97A
Pathway
Single-round viral replication assay
Decrease (50 %)
Approved
29769116
DrugRepV_6647Elvitegravir
Antiinfectives For Systemic Use
Acquired immunodeficiency syndrome
Human immunodeficiency virus
S119R
Pathway
Single-round viral replication assay
Decrease (50 %)
Approved
29769116
DrugRepV_6648Elvitegravir
Antiinfectives For Systemic Use
Acquired immunodeficiency syndrome
Human immunodeficiency virus
E138K
Pathway
Single-round viral replication assay
Decrease (50 %)
Approved
29769116
DrugRepV_6649Elvitegravir
Antiinfectives For Systemic Use
Acquired immunodeficiency syndrome
Human immunodeficiency virus
G140S
Pathway
Single-round viral replication assay
Decrease (50 %)
Approved
29769116
DrugRepV_6650Elvitegravir
Antiinfectives For Systemic Use
Acquired immunodeficiency syndrome
Human immunodeficiency virus
Q146L
Pathway
Single-round viral replication assay
Decrease (50 %)
Approved
29769116
DrugRepV_6651Elvitegravir
Antiinfectives For Systemic Use
Acquired immunodeficiency syndrome
Human immunodeficiency virus
Q146P
Pathway
Single-round viral replication assay
Decrease (50 %)
Approved
29769116
DrugRepV_6652Elvitegravir
Antiinfectives For Systemic Use
Acquired immunodeficiency syndrome
Human immunodeficiency virus
Q148H
Pathway
Single-round viral replication assay
Decrease (50 %)
Approved
29769116
DrugRepV_6653Elvitegravir
Antiinfectives For Systemic Use
Acquired immunodeficiency syndrome
Human immunodeficiency virus
Q148K
Pathway
Single-round viral replication assay
Decrease (50 %)
Approved
29769116
DrugRepV_6654Elvitegravir
Antiinfectives For Systemic Use
Acquired immunodeficiency syndrome
Human immunodeficiency virus
Q148R
Pathway
Single-round viral replication assay
Decrease (50 %)
Approved
29769116
DrugRepV_6655Elvitegravir
Antiinfectives For Systemic Use
Acquired immunodeficiency syndrome
Human immunodeficiency virus
S153Y
Pathway
Single-round viral replication assay
Decrease (50 %)
Approved
29769116
DrugRepV_6656Dolutegravir
Antiinfectives For Systemic Use
Acquired immunodeficiency syndrome
Human immunodeficiency virus
M50I
Pathway
Single-round viral replication assay
Decrease (50 %)
Approved
29769116
DrugRepV_6657Dolutegravir
Antiinfectives For Systemic Use
Acquired immunodeficiency syndrome
Human immunodeficiency virus
L74M
Pathway
Single-round viral replication assay
Decrease (50 %)
Approved
29769116
DrugRepV_6658Dolutegravir
Antiinfectives For Systemic Use
Acquired immunodeficiency syndrome
Human immunodeficiency virus
T97A
Pathway
Single-round viral replication assay
Decrease (50 %)
Approved
29769116
DrugRepV_6659Dolutegravir
Antiinfectives For Systemic Use
Acquired immunodeficiency syndrome
Human immunodeficiency virus
S119R
Pathway
Single-round viral replication assay
Decrease (50 %)
Approved
29769116
DrugRepV_6660Dolutegravir
Antiinfectives For Systemic Use
Acquired immunodeficiency syndrome
Human immunodeficiency virus
E138K
Pathway
Single-round viral replication assay
Decrease (50 %)
Approved
29769116
DrugRepV_6661Dolutegravir
Antiinfectives For Systemic Use
Acquired immunodeficiency syndrome
Human immunodeficiency virus
G140S
Pathway
Single-round viral replication assay
Decrease (50 %)
Approved
29769116
DrugRepV_6662Dolutegravir
Antiinfectives For Systemic Use
Acquired immunodeficiency syndrome
Human immunodeficiency virus
Q146L
Pathway
Single-round viral replication assay
Decrease (50 %)
Approved
29769116
DrugRepV_6663Dolutegravir
Antiinfectives For Systemic Use
Acquired immunodeficiency syndrome
Human immunodeficiency virus
Q146P
Pathway
Single-round viral replication assay
Decrease (50 %)
Approved
29769116
DrugRepV_6664Dolutegravir
Antiinfectives For Systemic Use
Acquired immunodeficiency syndrome
Human immunodeficiency virus
Q148H
Pathway
Single-round viral replication assay
Decrease (50 %)
Approved
29769116
DrugRepV_6665Dolutegravir
Antiinfectives For Systemic Use
Acquired immunodeficiency syndrome
Human immunodeficiency virus
Q148K
Pathway
Single-round viral replication assay
Decrease (50 %)
Approved
29769116
DrugRepV_6666Dolutegravir
Antiinfectives For Systemic Use
Acquired immunodeficiency syndrome
Human immunodeficiency virus
Q148R
Pathway
Single-round viral replication assay
Decrease (50 %)
Approved
29769116
DrugRepV_6667Dolutegravir
Antiinfectives For Systemic Use
Acquired immunodeficiency syndrome
Human immunodeficiency virus
S153Y
Pathway
Single-round viral replication assay
Decrease (50 %)
Approved
29769116
DrugRepV_6668Cabotegravir
Antiviral
Acquired immunodeficiency syndrome
Human immunodeficiency virus
M50I
Pathway
Single-round viral replication assay
Decrease (50 %)
Phase I
29769116
DrugRepV_6669Cabotegravir
Antiviral
Acquired immunodeficiency syndrome
Human immunodeficiency virus
L74M
Pathway
Single-round viral replication assay
Decrease (50 %)
Phase I
29769116
DrugRepV_6670Cabotegravir
Antiviral
Acquired immunodeficiency syndrome
Human immunodeficiency virus
T97A
Pathway
Single-round viral replication assay
Decrease (50 %)
Phase I
29769116
DrugRepV_6671Cabotegravir
Antiviral
Acquired immunodeficiency syndrome
Human immunodeficiency virus
S119R
Pathway
Single-round viral replication assay
Decrease (50 %)
Phase I
29769116
DrugRepV_6672Cabotegravir
Antiviral
Acquired immunodeficiency syndrome
Human immunodeficiency virus
E138K
Pathway
Single-round viral replication assay
Decrease (50 %)
Phase I
29769116
DrugRepV_6673Cabotegravir
Antiviral
Acquired immunodeficiency syndrome
Human immunodeficiency virus
G140S
Pathway
Single-round viral replication assay
Decrease (50 %)
Phase I
29769116
DrugRepV_6674Cabotegravir
Antiviral
Acquired immunodeficiency syndrome
Human immunodeficiency virus
Q146L
Pathway
Single-round viral replication assay
Decrease (50 %)
Phase I
29769116
DrugRepV_6675Cabotegravir
Antiviral
Acquired immunodeficiency syndrome
Human immunodeficiency virus
Q146P
Pathway
Single-round viral replication assay
Decrease (50 %)
Phase I
29769116
DrugRepV_6676Cabotegravir
Antiviral
Acquired immunodeficiency syndrome
Human immunodeficiency virus
Q148H
Pathway
Single-round viral replication assay
Decrease (50 %)
Phase I
29769116
DrugRepV_6677Cabotegravir
Antiviral
Acquired immunodeficiency syndrome
Human immunodeficiency virus
Q148K
Pathway
Single-round viral replication assay
Decrease (50 %)
Phase I
29769116
DrugRepV_6678Cabotegravir
Antiviral
Acquired immunodeficiency syndrome
Human immunodeficiency virus
Q148R
Pathway
Single-round viral replication assay
Decrease (50 %)
Phase I
29769116
DrugRepV_6679Cabotegravir
Antiviral
Acquired immunodeficiency syndrome
Human immunodeficiency virus
S153Y
Pathway
Single-round viral replication assay
Decrease (50 %)
Phase I
29769116
DrugRepV_6680Bictegravir
Antiinfectives For Systemic Use
Acquired immunodeficiency syndrome
Human immunodeficiency virus
M50I
Pathway
Single-round viral replication assay
Decrease (50 %)
Approved
29769116
DrugRepV_6681Bictegravir
Antiinfectives For Systemic Use
Acquired immunodeficiency syndrome
Human immunodeficiency virus
L74M
Pathway
Single-round viral replication assay
Decrease (50 %)
Approved
29769116
DrugRepV_6682Bictegravir
Antiinfectives For Systemic Use
Acquired immunodeficiency syndrome
Human immunodeficiency virus
T97A
Pathway
Single-round viral replication assay
Decrease (50 %)
Approved
29769116
DrugRepV_6683Bictegravir
Antiinfectives For Systemic Use
Acquired immunodeficiency syndrome
Human immunodeficiency virus
S119R
Pathway
Single-round viral replication assay
Decrease (50 %)
Approved
29769116
DrugRepV_6684Bictegravir
Antiinfectives For Systemic Use
Acquired immunodeficiency syndrome
Human immunodeficiency virus
E138K
Pathway
Single-round viral replication assay
Decrease (50 %)
Approved
29769116
DrugRepV_6685Bictegravir
Antiinfectives For Systemic Use
Acquired immunodeficiency syndrome
Human immunodeficiency virus
G140S
Pathway
Single-round viral replication assay
Decrease (50 %)
Approved
29769116
DrugRepV_6686Bictegravir
Antiinfectives For Systemic Use
Acquired immunodeficiency syndrome
Human immunodeficiency virus
Q146L
Pathway
Single-round viral replication assay
Decrease (50 %)
Approved
29769116
DrugRepV_6687Bictegravir
Antiinfectives For Systemic Use
Acquired immunodeficiency syndrome
Human immunodeficiency virus
Q146P
Pathway
Single-round viral replication assay
Decrease (50 %)
Approved
29769116
DrugRepV_6688Bictegravir
Antiinfectives For Systemic Use
Acquired immunodeficiency syndrome
Human immunodeficiency virus
Q148H
Pathway
Single-round viral replication assay
Decrease (50 %)
Approved
29769116
DrugRepV_6689Bictegravir
Antiinfectives For Systemic Use
Acquired immunodeficiency syndrome
Human immunodeficiency virus
Q148K
Pathway
Single-round viral replication assay
Decrease (50 %)
Approved
29769116
DrugRepV_6690Bictegravir
Antiinfectives For Systemic Use
Acquired immunodeficiency syndrome
Human immunodeficiency virus
Q148R
Pathway
Single-round viral replication assay
Decrease (50 %)
Approved
29769116
DrugRepV_6691Bictegravir
Antiinfectives For Systemic Use
Acquired immunodeficiency syndrome
Human immunodeficiency virus
S153Y
Pathway
Single-round viral replication assay
Decrease (50 %)
Approved
29769116
DrugRepV_6692Raltegravir
Antiinfectives For Systemic Use
Acquired immunodeficiency syndrome
Human immunodeficiency virus
G140A/Q148H
Pathway
Single-round viral replication assay
Decrease (50 %)
Approved
29769116
DrugRepV_6693Raltegravir
Antiinfectives For Systemic Use
Acquired immunodeficiency syndrome
Human immunodeficiency virus
Y143R/Q148H
Pathway
Single-round viral replication assay
Decrease (50 %)
Approved
29769116
DrugRepV_6694Raltegravir
Antiinfectives For Systemic Use
Acquired immunodeficiency syndrome
Human immunodeficiency virus
Q148H/N155H
Pathway
Single-round viral replication assay
Decrease (50 %)
Approved
29769116
DrugRepV_6695Raltegravir
Antiinfectives For Systemic Use
Acquired immunodeficiency syndrome
Human immunodeficiency virus
E138K/Q148K
Pathway
Single-round viral replication assay
Decrease (50 %)
Approved
29769116
DrugRepV_6696Raltegravir
Antiinfectives For Systemic Use
Acquired immunodeficiency syndrome
Human immunodeficiency virus
G140A/Q148K
Pathway
Single-round viral replication assay
Decrease (50 %)
Approved
29769116
DrugRepV_6697Raltegravir
Antiinfectives For Systemic Use
Acquired immunodeficiency syndrome
Human immunodeficiency virus
G140S/Q148K
Pathway
Single-round viral replication assay
Decrease (50 %)
Approved
29769116
DrugRepV_6698Raltegravir
Antiinfectives For Systemic Use
Acquired immunodeficiency syndrome
Human immunodeficiency virus
E138A/Q148R
Pathway
Single-round viral replication assay
Decrease (50 %)
Approved
29769116
DrugRepV_6699Raltegravir
Antiinfectives For Systemic Use
Acquired immunodeficiency syndrome
Human immunodeficiency virus
E138K/Q148R
Pathway
Single-round viral replication assay
Decrease (50 %)
Approved
29769116
DrugRepV_6700Raltegravir
Antiinfectives For Systemic Use
Acquired immunodeficiency syndrome
Human immunodeficiency virus
G140A/Q148R
Pathway
Single-round viral replication assay
Decrease (50 %)
Approved
29769116
DrugRepV_6701Raltegravir
Antiinfectives For Systemic Use
Acquired immunodeficiency syndrome
Human immunodeficiency virus
G140C/Q148R
Pathway
Single-round viral replication assay
Decrease (50 %)
Approved
29769116
DrugRepV_6702Raltegravir
Antiinfectives For Systemic Use
Acquired immunodeficiency syndrome
Human immunodeficiency virus
G140S/Q148R
Pathway
Single-round viral replication assay
Decrease (50 %)
Approved
29769116
DrugRepV_6703Raltegravir
Antiinfectives For Systemic Use
Acquired immunodeficiency syndrome
Human immunodeficiency virus
Q148R/N155H
Pathway
Single-round viral replication assay
Decrease (50 %)
Approved
29769116
DrugRepV_6704Elvitegravir
Antiinfectives For Systemic Use
Acquired immunodeficiency syndrome
Human immunodeficiency virus
G140A/Q148H
Pathway
Single-round viral replication assay
Decrease (50 %)
Approved
29769116
DrugRepV_6705Elvitegravir
Antiinfectives For Systemic Use
Acquired immunodeficiency syndrome
Human immunodeficiency virus
Y143R/Q148H
Pathway
Single-round viral replication assay
Decrease (50 %)
Approved
29769116
DrugRepV_6706Elvitegravir
Antiinfectives For Systemic Use
Acquired immunodeficiency syndrome
Human immunodeficiency virus
Q148H/N155H
Pathway
Single-round viral replication assay
Decrease (50 %)
Approved
29769116
DrugRepV_6707Elvitegravir
Antiinfectives For Systemic Use
Acquired immunodeficiency syndrome
Human immunodeficiency virus
E138K/Q148K
Pathway
Single-round viral replication assay
Decrease (50 %)
Approved
29769116
DrugRepV_6708Elvitegravir
Antiinfectives For Systemic Use
Acquired immunodeficiency syndrome
Human immunodeficiency virus
G140A/Q148K
Pathway
Single-round viral replication assay
Decrease (50 %)
Approved
29769116
DrugRepV_6709Elvitegravir
Antiinfectives For Systemic Use
Acquired immunodeficiency syndrome
Human immunodeficiency virus
G140S/Q148K
Pathway
Single-round viral replication assay
Decrease (50 %)
Approved
29769116
DrugRepV_6710Elvitegravir
Antiinfectives For Systemic Use
Acquired immunodeficiency syndrome
Human immunodeficiency virus
E138A/Q148R
Pathway
Single-round viral replication assay
Decrease (50 %)
Approved
29769116
DrugRepV_6711Elvitegravir
Antiinfectives For Systemic Use
Acquired immunodeficiency syndrome
Human immunodeficiency virus
E138K/Q148R
Pathway
Single-round viral replication assay
Decrease (50 %)
Approved
29769116
DrugRepV_6712Elvitegravir
Antiinfectives For Systemic Use
Acquired immunodeficiency syndrome
Human immunodeficiency virus
G140A/Q148R
Pathway
Single-round viral replication assay
Decrease (50 %)
Approved
29769116
DrugRepV_6713Elvitegravir
Antiinfectives For Systemic Use
Acquired immunodeficiency syndrome
Human immunodeficiency virus
G140C/Q148R
Pathway
Single-round viral replication assay
Decrease (50 %)
Approved
29769116
DrugRepV_6714Elvitegravir
Antiinfectives For Systemic Use
Acquired immunodeficiency syndrome
Human immunodeficiency virus
G140S/Q148R
Pathway
Single-round viral replication assay
Decrease (50 %)
Approved
29769116
DrugRepV_6715Elvitegravir
Antiinfectives For Systemic Use
Acquired immunodeficiency syndrome
Human immunodeficiency virus
Q148R/N155H
Pathway
Single-round viral replication assay
Decrease (50 %)
Approved
29769116
DrugRepV_6716Dolutegravir
Antiinfectives For Systemic Use
Acquired immunodeficiency syndrome
Human immunodeficiency virus
G140A/Q148H
Pathway
Single-round viral replication assay
Decrease (50 %)
Approved
29769116
DrugRepV_6717Dolutegravir
Antiinfectives For Systemic Use
Acquired immunodeficiency syndrome
Human immunodeficiency virus
Y143R/Q148H
Pathway
Single-round viral replication assay
Decrease (50 %)
Approved
29769116
DrugRepV_6718Dolutegravir
Antiinfectives For Systemic Use
Acquired immunodeficiency syndrome
Human immunodeficiency virus
Q148H/N155H
Pathway
Single-round viral replication assay
Decrease (50 %)
Approved
29769116
DrugRepV_6719Dolutegravir
Antiinfectives For Systemic Use
Acquired immunodeficiency syndrome
Human immunodeficiency virus
E138K/Q148K
Pathway
Single-round viral replication assay
Decrease (50 %)
Approved
29769116
DrugRepV_6720Dolutegravir
Antiinfectives For Systemic Use
Acquired immunodeficiency syndrome
Human immunodeficiency virus
G140A/Q148K
Pathway
Single-round viral replication assay
Decrease (50 %)
Approved
29769116
DrugRepV_6721Dolutegravir
Antiinfectives For Systemic Use
Acquired immunodeficiency syndrome
Human immunodeficiency virus
G140S/Q148K
Pathway
Single-round viral replication assay
Decrease (50 %)
Approved
29769116
DrugRepV_6722Dolutegravir
Antiinfectives For Systemic Use
Acquired immunodeficiency syndrome
Human immunodeficiency virus
E138A/Q148R
Pathway
Single-round viral replication assay
Decrease (50 %)
Approved
29769116
DrugRepV_6723Dolutegravir
Antiinfectives For Systemic Use
Acquired immunodeficiency syndrome
Human immunodeficiency virus
E138K/Q148R
Pathway
Single-round viral replication assay
Decrease (50 %)
Approved
29769116
DrugRepV_6724Dolutegravir
Antiinfectives For Systemic Use
Acquired immunodeficiency syndrome
Human immunodeficiency virus
G140A/Q148R
Pathway
Single-round viral replication assay
Decrease (50 %)
Approved
29769116
DrugRepV_6725Dolutegravir
Antiinfectives For Systemic Use
Acquired immunodeficiency syndrome
Human immunodeficiency virus
G140C/Q148R
Pathway
Single-round viral replication assay
Decrease (50 %)
Approved
29769116
DrugRepV_6726Dolutegravir
Antiinfectives For Systemic Use
Acquired immunodeficiency syndrome
Human immunodeficiency virus
G140S/Q148R
Pathway
Single-round viral replication assay
Decrease (50 %)
Approved
29769116
DrugRepV_6727Dolutegravir
Antiinfectives For Systemic Use
Acquired immunodeficiency syndrome
Human immunodeficiency virus
Q148R/N155H
Pathway
Single-round viral replication assay
Decrease (50 %)
Approved
29769116
DrugRepV_6728Cabotegravir
Antiviral
Acquired immunodeficiency syndrome
Human immunodeficiency virus
G140A/Q148H
Pathway
Single-round viral replication assay
Decrease (50 %)
Phase I
29769116
DrugRepV_6729Cabotegravir
Antiviral
Acquired immunodeficiency syndrome
Human immunodeficiency virus
Y143R/Q148H
Pathway
Single-round viral replication assay
Decrease (50 %)
Phase I
29769116
DrugRepV_6730Cabotegravir
Antiviral
Acquired immunodeficiency syndrome
Human immunodeficiency virus
Q148H/N155H
Pathway
Single-round viral replication assay
Decrease (50 %)
Phase I
29769116
DrugRepV_6731Cabotegravir
Antiviral
Acquired immunodeficiency syndrome
Human immunodeficiency virus
E138K/Q148K
Pathway
Single-round viral replication assay
Decrease (50 %)
Phase I
29769116
DrugRepV_6732Cabotegravir
Antiviral
Acquired immunodeficiency syndrome
Human immunodeficiency virus
G140A/Q148K
Pathway
Single-round viral replication assay
Decrease (50 %)
Phase I
29769116
DrugRepV_6733Cabotegravir
Antiviral
Acquired immunodeficiency syndrome
Human immunodeficiency virus
G140S/Q148K
Pathway
Single-round viral replication assay
Decrease (50 %)
Phase I
29769116
DrugRepV_6734Cabotegravir
Antiviral
Acquired immunodeficiency syndrome
Human immunodeficiency virus
E138A/Q148R
Pathway
Single-round viral replication assay
Decrease (50 %)
Phase I
29769116
DrugRepV_6735Cabotegravir
Antiviral
Acquired immunodeficiency syndrome
Human immunodeficiency virus
E138K/Q148R
Pathway
Single-round viral replication assay
Decrease (50 %)
Phase I
29769116
DrugRepV_6736Cabotegravir
Antiviral
Acquired immunodeficiency syndrome
Human immunodeficiency virus
G140A/Q148R
Pathway
Single-round viral replication assay
Decrease (50 %)
Phase I
29769116
DrugRepV_6737Cabotegravir
Antiviral
Acquired immunodeficiency syndrome
Human immunodeficiency virus
G140C/Q148R
Pathway
Single-round viral replication assay
Decrease (50 %)
Phase I
29769116
DrugRepV_6738Cabotegravir
Antiviral
Acquired immunodeficiency syndrome
Human immunodeficiency virus
G140S/Q148R
Pathway
Single-round viral replication assay
Decrease (50 %)
Phase I
29769116
DrugRepV_6739Cabotegravir
Antiviral
Acquired immunodeficiency syndrome
Human immunodeficiency virus
Q148R/N155H
Pathway
Single-round viral replication assay
Decrease (50 %)
Phase I
29769116
DrugRepV_6740Bictegravir
Antiinfectives For Systemic Use
Acquired immunodeficiency syndrome
Human immunodeficiency virus
G140A/Q148H
Pathway
Single-round viral replication assay
Decrease (50 %)
Approved
29769116
DrugRepV_6741Bictegravir
Antiinfectives For Systemic Use
Acquired immunodeficiency syndrome
Human immunodeficiency virus
Y143R/Q148H
Pathway
Single-round viral replication assay
Decrease (50 %)
Approved
29769116
DrugRepV_6742Bictegravir
Antiinfectives For Systemic Use
Acquired immunodeficiency syndrome
Human immunodeficiency virus
Q148H/N155H
Pathway
Single-round viral replication assay
Decrease (50 %)
Approved
29769116
DrugRepV_6743Bictegravir
Antiinfectives For Systemic Use
Acquired immunodeficiency syndrome
Human immunodeficiency virus
E138K/Q148K
Pathway
Single-round viral replication assay
Decrease (50 %)
Approved
29769116
DrugRepV_6744Bictegravir
Antiinfectives For Systemic Use
Acquired immunodeficiency syndrome
Human immunodeficiency virus
G140A/Q148K
Pathway
Single-round viral replication assay
Decrease (50 %)
Approved
29769116
DrugRepV_6745Bictegravir
Antiinfectives For Systemic Use
Acquired immunodeficiency syndrome
Human immunodeficiency virus
G140S/Q148K
Pathway
Single-round viral replication assay
Decrease (50 %)
Approved
29769116
DrugRepV_6746Bictegravir
Antiinfectives For Systemic Use
Acquired immunodeficiency syndrome
Human immunodeficiency virus
E138A/Q148R
Pathway
Single-round viral replication assay
Decrease (50 %)
Approved
29769116
DrugRepV_6747Bictegravir
Antiinfectives For Systemic Use
Acquired immunodeficiency syndrome
Human immunodeficiency virus
E138K/Q148R
Pathway
Single-round viral replication assay
Decrease (50 %)
Approved
29769116
DrugRepV_6748Bictegravir
Antiinfectives For Systemic Use
Acquired immunodeficiency syndrome
Human immunodeficiency virus
G140A/Q148R
Pathway
Single-round viral replication assay
Decrease (50 %)
Approved
29769116
DrugRepV_6749Bictegravir
Antiinfectives For Systemic Use
Acquired immunodeficiency syndrome
Human immunodeficiency virus
G140C/Q148R
Pathway
Single-round viral replication assay
Decrease (50 %)
Approved
29769116
DrugRepV_6750Bictegravir
Antiinfectives For Systemic Use
Acquired immunodeficiency syndrome
Human immunodeficiency virus
G140S/Q148R
Pathway
Single-round viral replication assay
Decrease (50 %)
Approved
29769116
DrugRepV_6751Bictegravir
Antiinfectives For Systemic Use
Acquired immunodeficiency syndrome
Human immunodeficiency virus
Q148R/N155H
Pathway
Single-round viral replication assay
Decrease (50 %)
Approved
29769116
DrugRepV_6752Raltegravir
Antiinfectives For Systemic Use
Acquired immunodeficiency syndrome
Human immunodeficiency virus
T66I/E157Q
Pathway
Single-round viral replication assay
Decrease (50 %)
Approved
29769116
DrugRepV_6753Raltegravir
Antiinfectives For Systemic Use
Acquired immunodeficiency syndrome
Human immunodeficiency virus
E92Q/N155H
Pathway
Single-round viral replication assay
Decrease (50 %)
Approved
29769116
DrugRepV_6754Raltegravir
Antiinfectives For Systemic Use
Acquired immunodeficiency syndrome
Human immunodeficiency virus
G140S/N155H
Pathway
Single-round viral replication assay
Decrease (50 %)
Approved
29769116
DrugRepV_6755Raltegravir
Antiinfectives For Systemic Use
Acquired immunodeficiency syndrome
Human immunodeficiency virus
Y143H/N155H
Pathway
Single-round viral replication assay
Decrease (50 %)
Approved
29769116
DrugRepV_6756Raltegravir
Antiinfectives For Systemic Use
Acquired immunodeficiency syndrome
Human immunodeficiency virus
Y143R/N155H
Pathway
Single-round viral replication assay
Decrease (50 %)
Approved
29769116
DrugRepV_6757Raltegravir
Antiinfectives For Systemic Use
Acquired immunodeficiency syndrome
Human immunodeficiency virus
N155H/G163R
Pathway
Single-round viral replication assay
Decrease (50 %)
Approved
29769116
DrugRepV_6758Elvitegravir
Antiinfectives For Systemic Use
Acquired immunodeficiency syndrome
Human immunodeficiency virus
T66I/E157Q
Pathway
Single-round viral replication assay
Decrease (50 %)
Approved
29769116
DrugRepV_6759Elvitegravir
Antiinfectives For Systemic Use
Acquired immunodeficiency syndrome
Human immunodeficiency virus
E92Q/N155H
Pathway
Single-round viral replication assay
Decrease (50 %)
Approved
29769116
DrugRepV_6760Elvitegravir
Antiinfectives For Systemic Use
Acquired immunodeficiency syndrome
Human immunodeficiency virus
G140S/N155H
Pathway
Single-round viral replication assay
Decrease (50 %)
Approved
29769116
DrugRepV_6761Elvitegravir
Antiinfectives For Systemic Use
Acquired immunodeficiency syndrome
Human immunodeficiency virus
Y143H/N155H
Pathway
Single-round viral replication assay
Decrease (50 %)
Approved
29769116
DrugRepV_6762Elvitegravir
Antiinfectives For Systemic Use
Acquired immunodeficiency syndrome
Human immunodeficiency virus
Y143R/N155H
Pathway
Single-round viral replication assay
Decrease (50 %)
Approved
29769116
DrugRepV_6763Elvitegravir
Antiinfectives For Systemic Use
Acquired immunodeficiency syndrome
Human immunodeficiency virus
N155H/G163R
Pathway
Single-round viral replication assay
Decrease (50 %)
Approved
29769116
DrugRepV_6764Dolutegravir
Antiinfectives For Systemic Use
Acquired immunodeficiency syndrome
Human immunodeficiency virus
T66I/E157Q
Pathway
Single-round viral replication assay
Decrease (50 %)
Approved
29769116
DrugRepV_6765Dolutegravir
Antiinfectives For Systemic Use
Acquired immunodeficiency syndrome
Human immunodeficiency virus
E92Q/N155H
Pathway
Single-round viral replication assay
Decrease (50 %)
Approved
29769116
DrugRepV_6766Dolutegravir
Antiinfectives For Systemic Use
Acquired immunodeficiency syndrome
Human immunodeficiency virus
G140S/N155H
Pathway
Single-round viral replication assay
Decrease (50 %)
Approved
29769116
DrugRepV_6767Dolutegravir
Antiinfectives For Systemic Use
Acquired immunodeficiency syndrome
Human immunodeficiency virus
Y143H/N155H
Pathway
Single-round viral replication assay
Decrease (50 %)
Approved
29769116
DrugRepV_6768Dolutegravir
Antiinfectives For Systemic Use
Acquired immunodeficiency syndrome
Human immunodeficiency virus
Y143R/N155H
Pathway
Single-round viral replication assay
Decrease (50 %)
Approved
29769116
DrugRepV_6769Dolutegravir
Antiinfectives For Systemic Use
Acquired immunodeficiency syndrome
Human immunodeficiency virus
N155H/G163R
Pathway
Single-round viral replication assay
Decrease (50 %)
Approved
29769116
DrugRepV_6770Cabotegravir
Antiviral
Acquired immunodeficiency syndrome
Human immunodeficiency virus
T66I/E157Q
Pathway
Single-round viral replication assay
Decrease (50 %)
Phase I
29769116
DrugRepV_6771Cabotegravir
Antiviral
Acquired immunodeficiency syndrome
Human immunodeficiency virus
E92Q/N155H
Pathway
Single-round viral replication assay
Decrease (50 %)
Phase I
29769116
DrugRepV_6772Cabotegravir
Antiviral
Acquired immunodeficiency syndrome
Human immunodeficiency virus
G140S/N155H
Pathway
Single-round viral replication assay
Decrease (50 %)
Phase I
29769116
DrugRepV_6773Cabotegravir
Antiviral
Acquired immunodeficiency syndrome
Human immunodeficiency virus
Y143H/N155H
Pathway
Single-round viral replication assay
Decrease (50 %)
Phase I
29769116
DrugRepV_6774Cabotegravir
Antiviral
Acquired immunodeficiency syndrome
Human immunodeficiency virus
Y143R/N155H
Pathway
Single-round viral replication assay
Decrease (50 %)
Phase I
29769116
DrugRepV_6775Cabotegravir
Antiviral
Acquired immunodeficiency syndrome
Human immunodeficiency virus
N155H/G163R
Pathway
Single-round viral replication assay
Decrease (50 %)
Phase I
29769116
DrugRepV_6776Bictegravir
Antiinfectives For Systemic Use
Acquired immunodeficiency syndrome
Human immunodeficiency virus
T66I/E157Q
Pathway
Single-round viral replication assay
Decrease (50 %)
Approved
29769116
DrugRepV_6777Bictegravir
Antiinfectives For Systemic Use
Acquired immunodeficiency syndrome
Human immunodeficiency virus
E92Q/N155H
Pathway
Single-round viral replication assay
Decrease (50 %)
Approved
29769116
DrugRepV_6778Bictegravir
Antiinfectives For Systemic Use
Acquired immunodeficiency syndrome
Human immunodeficiency virus
G140S/N155H
Pathway
Single-round viral replication assay
Decrease (50 %)
Approved
29769116
DrugRepV_6779Bictegravir
Antiinfectives For Systemic Use
Acquired immunodeficiency syndrome
Human immunodeficiency virus
Y143H/N155H
Pathway
Single-round viral replication assay
Decrease (50 %)
Approved
29769116
DrugRepV_6780Bictegravir
Antiinfectives For Systemic Use
Acquired immunodeficiency syndrome
Human immunodeficiency virus
Y143R/N155H
Pathway
Single-round viral replication assay
Decrease (50 %)
Approved
29769116
DrugRepV_6781Bictegravir
Antiinfectives For Systemic Use
Acquired immunodeficiency syndrome
Human immunodeficiency virus
N155H/G163R
Pathway
Single-round viral replication assay
Decrease (50 %)
Approved
29769116
DrugRepV_6782Raltegravir
Antiinfectives For Systemic Use
Acquired immunodeficiency syndrome
Human immunodeficiency virus
97A/Y143R/Q148H
Pathway
Single-round viral replication assay
Decrease (50 %)
Approved
29769116
DrugRepV_6783Raltegravir
Antiinfectives For Systemic Use
Acquired immunodeficiency syndrome
Human immunodeficiency virus
T97A/Q148H/N155H
Pathway
Single-round viral replication assay
Decrease (50 %)
Approved
29769116
DrugRepV_6784Raltegravir
Antiinfectives For Systemic Use
Acquired immunodeficiency syndrome
Human immunodeficiency virus
E138K/G140A/Q148K
Pathway
Single-round viral replication assay
Decrease (50 %)
Approved
29769116
DrugRepV_6785Raltegravir
Antiinfectives For Systemic Use
Acquired immunodeficiency syndrome
Human immunodeficiency virus
L74M/G140A/Q148R
Pathway
Single-round viral replication assay
Decrease (50 %)
Approved
29769116
DrugRepV_6786Raltegravir
Antiinfectives For Systemic Use
Acquired immunodeficiency syndrome
Human immunodeficiency virus
L74M/G140C/Q148R
Pathway
Single-round viral replication assay
Decrease (50 %)
Approved
29769116
DrugRepV_6787Raltegravir
Antiinfectives For Systemic Use
Acquired immunodeficiency syndrome
Human immunodeficiency virus
E138K/G140C/Q148R
Pathway
Single-round viral replication assay
Decrease (50 %)
Approved
29769116
DrugRepV_6788Raltegravir
Antiinfectives For Systemic Use
Acquired immunodeficiency syndrome
Human immunodeficiency virus
E138A/S147G/Q148R
Pathway
Single-round viral replication assay
Decrease (50 %)
Approved
29769116
DrugRepV_6789Elvitegravir
Antiinfectives For Systemic Use
Acquired immunodeficiency syndrome
Human immunodeficiency virus
97A/Y143R/Q148H
Pathway
Single-round viral replication assay
Decrease (50 %)
Approved
29769116
DrugRepV_6790Elvitegravir
Antiinfectives For Systemic Use
Acquired immunodeficiency syndrome
Human immunodeficiency virus
T97A/Q148H/N155H
Pathway
Single-round viral replication assay
Decrease (50 %)
Approved
29769116
DrugRepV_6791Elvitegravir
Antiinfectives For Systemic Use
Acquired immunodeficiency syndrome
Human immunodeficiency virus
E138K/G140A/Q148K
Pathway
Single-round viral replication assay
Decrease (50 %)
Approved
29769116
DrugRepV_6792Elvitegravir
Antiinfectives For Systemic Use
Acquired immunodeficiency syndrome
Human immunodeficiency virus
L74M/G140A/Q148R
Pathway
Single-round viral replication assay
Decrease (50 %)
Approved
29769116
DrugRepV_6793Elvitegravir
Antiinfectives For Systemic Use
Acquired immunodeficiency syndrome
Human immunodeficiency virus
L74M/G140C/Q148R
Pathway
Single-round viral replication assay
Decrease (50 %)
Approved
29769116
DrugRepV_6794Elvitegravir
Antiinfectives For Systemic Use
Acquired immunodeficiency syndrome
Human immunodeficiency virus
E138K/G140C/Q148R
Pathway
Single-round viral replication assay
Decrease (50 %)
Approved
29769116
DrugRepV_6795Elvitegravir
Antiinfectives For Systemic Use
Acquired immunodeficiency syndrome
Human immunodeficiency virus
E138A/S147G/Q148R
Pathway
Single-round viral replication assay
Decrease (50 %)
Approved
29769116
DrugRepV_6796Dolutegravir
Antiinfectives For Systemic Use
Acquired immunodeficiency syndrome
Human immunodeficiency virus
97A/Y143R/Q148H
Pathway
Single-round viral replication assay
Decrease (50 %)
Approved
29769116
DrugRepV_6797Dolutegravir
Antiinfectives For Systemic Use
Acquired immunodeficiency syndrome
Human immunodeficiency virus
T97A/Q148H/N155H
Pathway
Single-round viral replication assay
Decrease (50 %)
Approved
29769116
DrugRepV_6798Dolutegravir
Antiinfectives For Systemic Use
Acquired immunodeficiency syndrome
Human immunodeficiency virus
E138K/G140A/Q148K
Pathway
Single-round viral replication assay
Decrease (50 %)
Approved
29769116
DrugRepV_6799Dolutegravir
Antiinfectives For Systemic Use
Acquired immunodeficiency syndrome
Human immunodeficiency virus
L74M/G140A/Q148R
Pathway
Single-round viral replication assay
Decrease (50 %)
Approved
29769116
DrugRepV_6800Dolutegravir
Antiinfectives For Systemic Use
Acquired immunodeficiency syndrome
Human immunodeficiency virus
L74M/G140C/Q148R
Pathway
Single-round viral replication assay
Decrease (50 %)
Approved
29769116
DrugRepV_6801Dolutegravir
Antiinfectives For Systemic Use
Acquired immunodeficiency syndrome
Human immunodeficiency virus
E138K/G140C/Q148R
Pathway
Single-round viral replication assay
Decrease (50 %)
Approved
29769116
DrugRepV_6802Dolutegravir
Antiinfectives For Systemic Use
Acquired immunodeficiency syndrome
Human immunodeficiency virus
E138A/S147G/Q148R
Pathway
Single-round viral replication assay
Decrease (50 %)
Approved
29769116
DrugRepV_6803Cabotegravir
Antiviral
Acquired immunodeficiency syndrome
Human immunodeficiency virus
97A/Y143R/Q148H
Pathway
Single-round viral replication assay
Decrease (50 %)
Phase I
29769116
DrugRepV_6804Cabotegravir
Antiviral
Acquired immunodeficiency syndrome
Human immunodeficiency virus
T97A/Q148H/N155H
Pathway
Single-round viral replication assay
Decrease (50 %)
Phase I
29769116
DrugRepV_6805Cabotegravir
Antiviral
Acquired immunodeficiency syndrome
Human immunodeficiency virus
E138K/G140A/Q148K
Pathway
Single-round viral replication assay
Decrease (50 %)
Phase I
29769116
DrugRepV_6806Cabotegravir
Antiviral
Acquired immunodeficiency syndrome
Human immunodeficiency virus
L74M/G140A/Q148R
Pathway
Single-round viral replication assay
Decrease (50 %)
Phase I
29769116
DrugRepV_6807Cabotegravir
Antiviral
Acquired immunodeficiency syndrome
Human immunodeficiency virus
L74M/G140C/Q148R
Pathway
Single-round viral replication assay
Decrease (50 %)
Phase I
29769116
DrugRepV_6808Cabotegravir
Antiviral
Acquired immunodeficiency syndrome
Human immunodeficiency virus
E138K/G140C/Q148R
Pathway
Single-round viral replication assay
Decrease (50 %)
Phase I
29769116
DrugRepV_6809Cabotegravir
Antiviral
Acquired immunodeficiency syndrome
Human immunodeficiency virus
E138A/S147G/Q148R
Pathway
Single-round viral replication assay
Decrease (50 %)
Phase I
29769116
DrugRepV_6810Bictegravir
Antiinfectives For Systemic Use
Acquired immunodeficiency syndrome
Human immunodeficiency virus
97A/Y143R/Q148H
Pathway
Single-round viral replication assay
Decrease (50 %)
Approved
29769116
DrugRepV_6811Bictegravir
Antiinfectives For Systemic Use
Acquired immunodeficiency syndrome
Human immunodeficiency virus
T97A/Q148H/N155H
Pathway
Single-round viral replication assay
Decrease (50 %)
Approved
29769116
DrugRepV_6812Bictegravir
Antiinfectives For Systemic Use
Acquired immunodeficiency syndrome
Human immunodeficiency virus
E138K/G140A/Q148K
Pathway
Single-round viral replication assay
Decrease (50 %)
Approved
29769116
DrugRepV_6813Bictegravir
Antiinfectives For Systemic Use
Acquired immunodeficiency syndrome
Human immunodeficiency virus
L74M/G140A/Q148R
Pathway
Single-round viral replication assay
Decrease (50 %)
Approved
29769116
DrugRepV_6814Bictegravir
Antiinfectives For Systemic Use
Acquired immunodeficiency syndrome
Human immunodeficiency virus
L74M/G140C/Q148R
Pathway
Single-round viral replication assay
Decrease (50 %)
Approved
29769116
DrugRepV_6815Bictegravir
Antiinfectives For Systemic Use
Acquired immunodeficiency syndrome
Human immunodeficiency virus
E138K/G140C/Q148R
Pathway
Single-round viral replication assay
Decrease (50 %)
Approved
29769116
DrugRepV_6816Bictegravir
Antiinfectives For Systemic Use
Acquired immunodeficiency syndrome
Human immunodeficiency virus
E138A/S147G/Q148R
Pathway
Single-round viral replication assay
Decrease (50 %)
Approved
29769116
DrugRepV_6817Raltegravir
Antiinfectives For Systemic Use
Acquired immunodeficiency syndrome
Human immunodeficiency virus
T66I/T97A/E157Q
Pathway
Single-round viral replication assay
Decrease (50 %)
Approved
29769116
DrugRepV_6818Raltegravir
Antiinfectives For Systemic Use
Acquired immunodeficiency syndrome
Human immunodeficiency virus
T97A/Y143R/N155H
Pathway
Single-round viral replication assay
Decrease (50 %)
Approved
29769116
DrugRepV_6819Raltegravir
Antiinfectives For Systemic Use
Acquired immunodeficiency syndrome
Human immunodeficiency virus
G140S/Y143R/N155H
Pathway
Single-round viral replication assay
Decrease (50 %)
Approved
29769116
DrugRepV_6820Raltegravir
Antiinfectives For Systemic Use
Acquired immunodeficiency syndrome
Human immunodeficiency virus
E92Q/N155H/G163R
Pathway
Single-round viral replication assay
Decrease (50 %)
Approved
29769116
DrugRepV_6821Elvitegravir
Antiinfectives For Systemic Use
Acquired immunodeficiency syndrome
Human immunodeficiency virus
T66I/T97A/E157Q
Pathway
Single-round viral replication assay
Decrease (50 %)
Approved
29769116
DrugRepV_6822Elvitegravir
Antiinfectives For Systemic Use
Acquired immunodeficiency syndrome
Human immunodeficiency virus
T97A/Y143R/N155H
Pathway
Single-round viral replication assay
Decrease (50 %)
Approved
29769116
DrugRepV_6823Elvitegravir
Antiinfectives For Systemic Use
Acquired immunodeficiency syndrome
Human immunodeficiency virus
G140S/Y143R/N155H
Pathway
Single-round viral replication assay
Decrease (50 %)
Approved
29769116
DrugRepV_6824Elvitegravir
Antiinfectives For Systemic Use
Acquired immunodeficiency syndrome
Human immunodeficiency virus
E92Q/N155H/G163R
Pathway
Single-round viral replication assay
Decrease (50 %)
Approved
29769116
DrugRepV_6825Dolutegravir
Antiinfectives For Systemic Use
Acquired immunodeficiency syndrome
Human immunodeficiency virus
T66I/T97A/E157Q
Pathway
Single-round viral replication assay
Decrease (50 %)
Approved
29769116
DrugRepV_6826Dolutegravir
Antiinfectives For Systemic Use
Acquired immunodeficiency syndrome
Human immunodeficiency virus
T97A/Y143R/N155H
Pathway
Single-round viral replication assay
Decrease (50 %)
Approved
29769116
DrugRepV_6827Dolutegravir
Antiinfectives For Systemic Use
Acquired immunodeficiency syndrome
Human immunodeficiency virus
G140S/Y143R/N155H
Pathway
Single-round viral replication assay
Decrease (50 %)
Approved
29769116
DrugRepV_6828Dolutegravir
Antiinfectives For Systemic Use
Acquired immunodeficiency syndrome
Human immunodeficiency virus
E92Q/N155H/G163R
Pathway
Single-round viral replication assay
Decrease (50 %)
Approved
29769116
DrugRepV_6829Cabotegravir
Antiviral
Acquired immunodeficiency syndrome
Human immunodeficiency virus
T66I/T97A/E157Q
Pathway
Single-round viral replication assay
Decrease (50 %)
Phase I
29769116
DrugRepV_6830Cabotegravir
Antiviral
Acquired immunodeficiency syndrome
Human immunodeficiency virus
T97A/Y143R/N155H
Pathway
Single-round viral replication assay
Decrease (50 %)
Phase I
29769116
DrugRepV_6831Cabotegravir
Antiviral
Acquired immunodeficiency syndrome
Human immunodeficiency virus
G140S/Y143R/N155H
Pathway
Single-round viral replication assay
Decrease (50 %)
Phase I
29769116
DrugRepV_6832Cabotegravir
Antiviral
Acquired immunodeficiency syndrome
Human immunodeficiency virus
E92Q/N155H/G163R
Pathway
Single-round viral replication assay
Decrease (50 %)
Phase I
29769116
DrugRepV_6833Bictegravir
Antiinfectives For Systemic Use
Acquired immunodeficiency syndrome
Human immunodeficiency virus
T66I/T97A/E157Q
Pathway
Single-round viral replication assay
Decrease (50 %)
Approved
29769116
DrugRepV_6834Bictegravir
Antiinfectives For Systemic Use
Acquired immunodeficiency syndrome
Human immunodeficiency virus
T97A/Y143R/N155H
Pathway
Single-round viral replication assay
Decrease (50 %)
Approved
29769116
DrugRepV_6835Bictegravir
Antiinfectives For Systemic Use
Acquired immunodeficiency syndrome
Human immunodeficiency virus
G140S/Y143R/N155H
Pathway
Single-round viral replication assay
Decrease (50 %)
Approved
29769116
DrugRepV_6836Bictegravir
Antiinfectives For Systemic Use
Acquired immunodeficiency syndrome
Human immunodeficiency virus
E92Q/N155H/G163R
Pathway
Single-round viral replication assay
Decrease (50 %)
Approved
29769116
DrugRepV_6837Raltegravir
Antiinfectives For Systemic Use
Acquired immunodeficiency syndrome
Human immunodeficiency virus
T97A/G140S/Q148H
Pathway
Single-round viral replication assay
Decrease (50 %)
Approved
29769116
DrugRepV_6838Raltegravir
Antiinfectives For Systemic Use
Acquired immunodeficiency syndrome
Human immunodeficiency virus
E138A/G140S/Q148H
Pathway
Single-round viral replication assay
Decrease (50 %)
Approved
29769116
DrugRepV_6839Raltegravir
Antiinfectives For Systemic Use
Acquired immunodeficiency syndrome
Human immunodeficiency virus
E138K/G140S/Q148H
Pathway
Single-round viral replication assay
Decrease (50 %)
Approved
29769116
DrugRepV_6840Raltegravir
Antiinfectives For Systemic Use
Acquired immunodeficiency syndrome
Human immunodeficiency virus
G140S/Y143R/Q148H
Pathway
Single-round viral replication assay
Decrease (50 %)
Approved
29769116
DrugRepV_6841Raltegravir
Antiinfectives For Systemic Use
Acquired immunodeficiency syndrome
Human immunodeficiency virus
G140S/Q148H/N155H
Pathway
Single-round viral replication assay
Decrease (50 %)
Approved
29769116
DrugRepV_6842Raltegravir
Antiinfectives For Systemic Use
Acquired immunodeficiency syndrome
Human immunodeficiency virus
G140S/Q148H/G163K
Pathway
Single-round viral replication assay
Decrease (50 %)
Approved
29769116
DrugRepV_6843Elvitegravir
Antiinfectives For Systemic Use
Acquired immunodeficiency syndrome
Human immunodeficiency virus
T97A/G140S/Q148H
Pathway
Single-round viral replication assay
Decrease (50 %)
Approved
29769116
DrugRepV_6844Elvitegravir
Antiinfectives For Systemic Use
Acquired immunodeficiency syndrome
Human immunodeficiency virus
E138A/G140S/Q148H
Pathway
Single-round viral replication assay
Decrease (50 %)
Approved
29769116
DrugRepV_6845Elvitegravir
Antiinfectives For Systemic Use
Acquired immunodeficiency syndrome
Human immunodeficiency virus
E138K/G140S/Q148H
Pathway
Single-round viral replication assay
Decrease (50 %)
Approved
29769116
DrugRepV_6846Elvitegravir
Antiinfectives For Systemic Use
Acquired immunodeficiency syndrome
Human immunodeficiency virus
G140S/Y143R/Q148H
Pathway
Single-round viral replication assay
Decrease (50 %)
Approved
29769116
DrugRepV_6847Elvitegravir
Antiinfectives For Systemic Use
Acquired immunodeficiency syndrome
Human immunodeficiency virus
G140S/Q148H/N155H
Pathway
Single-round viral replication assay
Decrease (50 %)
Approved
29769116
DrugRepV_6848Elvitegravir
Antiinfectives For Systemic Use
Acquired immunodeficiency syndrome
Human immunodeficiency virus
G140S/Q148H/G163K
Pathway
Single-round viral replication assay
Decrease (50 %)
Approved
29769116
DrugRepV_6849Dolutegravir
Antiinfectives For Systemic Use
Acquired immunodeficiency syndrome
Human immunodeficiency virus
T97A/G140S/Q148H
Pathway
Single-round viral replication assay
Decrease (50 %)
Approved
29769116
DrugRepV_6850Dolutegravir
Antiinfectives For Systemic Use
Acquired immunodeficiency syndrome
Human immunodeficiency virus
E138A/G140S/Q148H
Pathway
Single-round viral replication assay
Decrease (50 %)
Approved
29769116
DrugRepV_6851Dolutegravir
Antiinfectives For Systemic Use
Acquired immunodeficiency syndrome
Human immunodeficiency virus
E138K/G140S/Q148H
Pathway
Single-round viral replication assay
Decrease (50 %)
Approved
29769116
DrugRepV_6852Dolutegravir
Antiinfectives For Systemic Use
Acquired immunodeficiency syndrome
Human immunodeficiency virus
G140S/Y143R/Q148H
Pathway
Single-round viral replication assay
Decrease (50 %)
Approved
29769116
DrugRepV_6853Dolutegravir
Antiinfectives For Systemic Use
Acquired immunodeficiency syndrome
Human immunodeficiency virus
G140S/Q148H/N155H
Pathway
Single-round viral replication assay
Decrease (50 %)
Approved
29769116
DrugRepV_6854Dolutegravir
Antiinfectives For Systemic Use
Acquired immunodeficiency syndrome
Human immunodeficiency virus
G140S/Q148H/G163K
Pathway
Single-round viral replication assay
Decrease (50 %)
Approved
29769116
DrugRepV_6855Cabotegravir
Antiviral
Acquired immunodeficiency syndrome
Human immunodeficiency virus
T97A/G140S/Q148H
Pathway
Single-round viral replication assay
Decrease (50 %)
Phase I
29769116
DrugRepV_6856Cabotegravir
Antiviral
Acquired immunodeficiency syndrome
Human immunodeficiency virus
E138A/G140S/Q148H
Pathway
Single-round viral replication assay
Decrease (50 %)
Phase I
29769116
DrugRepV_6857Cabotegravir
Antiviral
Acquired immunodeficiency syndrome
Human immunodeficiency virus
E138K/G140S/Q148H
Pathway
Single-round viral replication assay
Decrease (50 %)
Phase I
29769116
DrugRepV_6858Cabotegravir
Antiviral
Acquired immunodeficiency syndrome
Human immunodeficiency virus
G140S/Y143R/Q148H
Pathway
Single-round viral replication assay
Decrease (50 %)
Phase I
29769116
DrugRepV_6859Cabotegravir
Antiviral
Acquired immunodeficiency syndrome
Human immunodeficiency virus
G140S/Q148H/N155H
Pathway
Single-round viral replication assay
Decrease (50 %)
Phase I
29769116
DrugRepV_6860Cabotegravir
Antiviral
Acquired immunodeficiency syndrome
Human immunodeficiency virus
G140S/Q148H/G163K
Pathway
Single-round viral replication assay
Decrease (50 %)
Phase I
29769116
DrugRepV_6861Bictegravir
Antiinfectives For Systemic Use
Acquired immunodeficiency syndrome
Human immunodeficiency virus
T97A/G140S/Q148H
Pathway
Single-round viral replication assay
Decrease (50 %)
Approved
29769116
DrugRepV_6862Bictegravir
Antiinfectives For Systemic Use
Acquired immunodeficiency syndrome
Human immunodeficiency virus
E138A/G140S/Q148H
Pathway
Single-round viral replication assay
Decrease (50 %)
Approved
29769116
DrugRepV_6863Bictegravir
Antiinfectives For Systemic Use
Acquired immunodeficiency syndrome
Human immunodeficiency virus
E138K/G140S/Q148H
Pathway
Single-round viral replication assay
Decrease (50 %)
Approved
29769116
DrugRepV_6864Bictegravir
Antiinfectives For Systemic Use
Acquired immunodeficiency syndrome
Human immunodeficiency virus
G140S/Y143R/Q148H
Pathway
Single-round viral replication assay
Decrease (50 %)
Approved
29769116
DrugRepV_6865Bictegravir
Antiinfectives For Systemic Use
Acquired immunodeficiency syndrome
Human immunodeficiency virus
G140S/Q148H/N155H
Pathway
Single-round viral replication assay
Decrease (50 %)
Approved
29769116
DrugRepV_6866Bictegravir
Antiinfectives For Systemic Use
Acquired immunodeficiency syndrome
Human immunodeficiency virus
G140S/Q148H/G163K
Pathway
Single-round viral replication assay
Decrease (50 %)
Approved
29769116