DrugRepV_6577 | Raltegravir | Antiinfectives For Systemic Use | Acquired immunodeficiency syndrome | Human immunodeficiency virus | WT | | Single-round viral replication assay | Decrease (50 %) | Approved | 29769116 |
DrugRepV_6578 | Raltegravir | Antiinfectives For Systemic Use | Acquired immunodeficiency syndrome | Human immunodeficiency virus | Y143R (RAL) | | Single-round viral replication assay | Decrease (50 %) | Approved | 29769116 |
DrugRepV_6579 | Raltegravir | Antiinfectives For Systemic Use | Acquired immunodeficiency syndrome | Human immunodeficiency virus | N155H(RAL) | | Single-round viral replication assay | Decrease (50 %) | Approved | 29769116 |
DrugRepV_6580 | Raltegravir | Antiinfectives For Systemic Use | Acquired immunodeficiency syndrome | Human immunodeficiency virus | G140S/Q148H (RAL) | | Single-round viral replication assay | Decrease (50 %) | Approved | 29769116 |
DrugRepV_6581 | Raltegravir | Antiinfectives For Systemic Use | Acquired immunodeficiency syndrome | Human immunodeficiency virus | T661(EVG) | | Single-round viral replication assay | Decrease (50 %) | Approved | 29769116 |
DrugRepV_6582 | Raltegravir | Antiinfectives For Systemic Use | Acquired immunodeficiency syndrome | Human immunodeficiency virus | E92Q (EVG) | | Single-round viral replication assay | Decrease (50 %) | Approved | 29769116 |
DrugRepV_6583 | Raltegravir | Antiinfectives For Systemic Use | Acquired immunodeficiency syndrome | Human immunodeficiency virus | H51Y (DTG) | | Single-round viral replication assay | Decrease (50 %) | Approved | 29769116 |
DrugRepV_6584 | Raltegravir | Antiinfectives For Systemic Use | Acquired immunodeficiency syndrome | Human immunodeficiency virus | G118R (DTG) | | Single-round viral replication assay | Decrease (50 %) | Approved | 29769116 |
DrugRepV_6585 | Raltegravir | Antiinfectives For Systemic Use | Acquired immunodeficiency syndrome | Human immunodeficiency virus | R263K (DTG) | | Single-round viral replication assay | Decrease (50 %) | Approved | 29769116 |
DrugRepV_6586 | Raltegravir | Antiinfectives For Systemic Use | Acquired immunodeficiency syndrome | Human immunodeficiency virus | H51Y/R263K (DTG) | | Single-round viral replication assay | Decrease (50 %) | Approved | 29769116 |
DrugRepV_6587 | Raltegravir | Antiinfectives For Systemic Use | Acquired immunodeficiency syndrome | Human immunodeficiency virus | E138K/R263K (DTG) | | Single-round viral replication assay | Decrease (50 %) | Approved | 29769116 |
DrugRepV_6588 | Elvitegravir | Antiinfectives For Systemic Use | Acquired immunodeficiency syndrome | Human immunodeficiency virus | WT | | Single-round viral replication assay | Decrease (50 %) | Approved | 29769116 |
DrugRepV_6589 | Elvitegravir | Antiinfectives For Systemic Use | Acquired immunodeficiency syndrome | Human immunodeficiency virus | Y143R (RAL) | | Single-round viral replication assay | Decrease (50 %) | Approved | 29769116 |
DrugRepV_6590 | Elvitegravir | Antiinfectives For Systemic Use | Acquired immunodeficiency syndrome | Human immunodeficiency virus | N155H(RAL) | | Single-round viral replication assay | Decrease (50 %) | Approved | 29769116 |
DrugRepV_6591 | Elvitegravir | Antiinfectives For Systemic Use | Acquired immunodeficiency syndrome | Human immunodeficiency virus | G140S/Q148H (RAL) | | Single-round viral replication assay | Decrease (50 %) | Approved | 29769116 |
DrugRepV_6592 | Elvitegravir | Antiinfectives For Systemic Use | Acquired immunodeficiency syndrome | Human immunodeficiency virus | T661(EVG) | | Single-round viral replication assay | Decrease (50 %) | Approved | 29769116 |
DrugRepV_6593 | Elvitegravir | Antiinfectives For Systemic Use | Acquired immunodeficiency syndrome | Human immunodeficiency virus | E92Q (EVG) | | Single-round viral replication assay | Decrease (50 %) | Approved | 29769116 |
DrugRepV_6594 | Elvitegravir | Antiinfectives For Systemic Use | Acquired immunodeficiency syndrome | Human immunodeficiency virus | H51Y (DTG) | | Single-round viral replication assay | Decrease (50 %) | Approved | 29769116 |
DrugRepV_6595 | Elvitegravir | Antiinfectives For Systemic Use | Acquired immunodeficiency syndrome | Human immunodeficiency virus | G118R (DTG) | | Single-round viral replication assay | Decrease (50 %) | Approved | 29769116 |
DrugRepV_6596 | Elvitegravir | Antiinfectives For Systemic Use | Acquired immunodeficiency syndrome | Human immunodeficiency virus | R263K (DTG) | | Single-round viral replication assay | Decrease (50 %) | Approved | 29769116 |
DrugRepV_6597 | Elvitegravir | Antiinfectives For Systemic Use | Acquired immunodeficiency syndrome | Human immunodeficiency virus | H51Y/R263K (DTG) | | Single-round viral replication assay | Decrease (50 %) | Approved | 29769116 |
DrugRepV_6598 | Elvitegravir | Antiinfectives For Systemic Use | Acquired immunodeficiency syndrome | Human immunodeficiency virus | E138K/R263K (DTG) | | Single-round viral replication assay | Decrease (50 %) | Approved | 29769116 |
DrugRepV_6599 | Dolutegravir | Antiinfectives For Systemic Use | Acquired immunodeficiency syndrome | Human immunodeficiency virus | WT | | Single-round viral replication assay | Decrease (50 %) | Approved | 29769116 |
DrugRepV_6600 | Dolutegravir | Antiinfectives For Systemic Use | Acquired immunodeficiency syndrome | Human immunodeficiency virus | Y143R (RAL) | | Single-round viral replication assay | Decrease (50 %) | Approved | 29769116 |
DrugRepV_6601 | Dolutegravir | Antiinfectives For Systemic Use | Acquired immunodeficiency syndrome | Human immunodeficiency virus | N155H(RAL) | | Single-round viral replication assay | Decrease (50 %) | Approved | 29769116 |
DrugRepV_6602 | Dolutegravir | Antiinfectives For Systemic Use | Acquired immunodeficiency syndrome | Human immunodeficiency virus | G140S/Q148H (RAL) | | Single-round viral replication assay | Decrease (50 %) | Approved | 29769116 |
DrugRepV_6603 | Dolutegravir | Antiinfectives For Systemic Use | Acquired immunodeficiency syndrome | Human immunodeficiency virus | T661(EVG) | | Single-round viral replication assay | Decrease (50 %) | Approved | 29769116 |
DrugRepV_6604 | Dolutegravir | Antiinfectives For Systemic Use | Acquired immunodeficiency syndrome | Human immunodeficiency virus | E92Q (EVG) | | Single-round viral replication assay | Decrease (50 %) | Approved | 29769116 |
DrugRepV_6605 | Dolutegravir | Antiinfectives For Systemic Use | Acquired immunodeficiency syndrome | Human immunodeficiency virus | H51Y (DTG) | | Single-round viral replication assay | Decrease (50 %) | Approved | 29769116 |
DrugRepV_6606 | Dolutegravir | Antiinfectives For Systemic Use | Acquired immunodeficiency syndrome | Human immunodeficiency virus | G118R (DTG) | | Single-round viral replication assay | Decrease (50 %) | Approved | 29769116 |
DrugRepV_6607 | Dolutegravir | Antiinfectives For Systemic Use | Acquired immunodeficiency syndrome | Human immunodeficiency virus | R263K (DTG) | | Single-round viral replication assay | Decrease (50 %) | Approved | 29769116 |
DrugRepV_6608 | Dolutegravir | Antiinfectives For Systemic Use | Acquired immunodeficiency syndrome | Human immunodeficiency virus | H51Y/R263K (DTG) | | Single-round viral replication assay | Decrease (50 %) | Approved | 29769116 |
DrugRepV_6609 | Dolutegravir | Antiinfectives For Systemic Use | Acquired immunodeficiency syndrome | Human immunodeficiency virus | E138K/R263K (DTG) | | Single-round viral replication assay | Decrease (50 %) | Approved | 29769116 |
DrugRepV_6610 | Cabotegravir | Antiviral | Acquired immunodeficiency syndrome | Human immunodeficiency virus | WT | | Single-round viral replication assay | Decrease (50 %) | Phase I | 29769116 |
DrugRepV_6611 | Cabotegravir | Antiviral | Acquired immunodeficiency syndrome | Human immunodeficiency virus | Y143R (RAL) | | Single-round viral replication assay | Decrease (50 %) | Phase I | 29769116 |
DrugRepV_6612 | Cabotegravir | Antiviral | Acquired immunodeficiency syndrome | Human immunodeficiency virus | N155H(RAL) | | Single-round viral replication assay | Decrease (50 %) | Phase I | 29769116 |
DrugRepV_6613 | Cabotegravir | Antiviral | Acquired immunodeficiency syndrome | Human immunodeficiency virus | G140S/Q148H (RAL) | | Single-round viral replication assay | Decrease (50 %) | Phase I | 29769116 |
DrugRepV_6614 | Cabotegravir | Antiviral | Acquired immunodeficiency syndrome | Human immunodeficiency virus | T661(EVG) | | Single-round viral replication assay | Decrease (50 %) | Phase I | 29769116 |
DrugRepV_6615 | Cabotegravir | Antiviral | Acquired immunodeficiency syndrome | Human immunodeficiency virus | E92Q (EVG) | | Single-round viral replication assay | Decrease (50 %) | Phase I | 29769116 |
DrugRepV_6616 | Cabotegravir | Antiviral | Acquired immunodeficiency syndrome | Human immunodeficiency virus | H51Y (DTG) | | Single-round viral replication assay | Decrease (50 %) | Phase I | 29769116 |
DrugRepV_6617 | Cabotegravir | Antiviral | Acquired immunodeficiency syndrome | Human immunodeficiency virus | G118R (DTG) | | Single-round viral replication assay | Decrease (50 %) | Phase I | 29769116 |
DrugRepV_6618 | Cabotegravir | Antiviral | Acquired immunodeficiency syndrome | Human immunodeficiency virus | R263K (DTG) | | Single-round viral replication assay | Decrease (50 %) | Phase I | 29769116 |
DrugRepV_6619 | Cabotegravir | Antiviral | Acquired immunodeficiency syndrome | Human immunodeficiency virus | H51Y/R263K (DTG) | | Single-round viral replication assay | Decrease (50 %) | Phase I | 29769116 |
DrugRepV_6620 | Cabotegravir | Antiviral | Acquired immunodeficiency syndrome | Human immunodeficiency virus | E138K/R263K (DTG) | | Single-round viral replication assay | Decrease (50 %) | Phase I | 29769116 |
DrugRepV_6621 | Bictegravir | Antiinfectives For Systemic Use | Acquired immunodeficiency syndrome | Human immunodeficiency virus | WT | | Single-round viral replication assay | Decrease (50 %) | Approved | 29769116 |
DrugRepV_6622 | Bictegravir | Antiinfectives For Systemic Use | Acquired immunodeficiency syndrome | Human immunodeficiency virus | Y143R (RAL) | | Single-round viral replication assay | Decrease (50 %) | Approved | 29769116 |
DrugRepV_6623 | Bictegravir | Antiinfectives For Systemic Use | Acquired immunodeficiency syndrome | Human immunodeficiency virus | N155H(RAL) | | Single-round viral replication assay | Decrease (50 %) | Approved | 29769116 |
DrugRepV_6624 | Bictegravir | Antiinfectives For Systemic Use | Acquired immunodeficiency syndrome | Human immunodeficiency virus | G140S/Q148H (RAL) | | Single-round viral replication assay | Decrease (50 %) | Approved | 29769116 |
DrugRepV_6625 | Bictegravir | Antiinfectives For Systemic Use | Acquired immunodeficiency syndrome | Human immunodeficiency virus | T661(EVG) | | Single-round viral replication assay | Decrease (50 %) | Approved | 29769116 |
DrugRepV_6626 | Bictegravir | Antiinfectives For Systemic Use | Acquired immunodeficiency syndrome | Human immunodeficiency virus | E92Q (EVG) | | Single-round viral replication assay | Decrease (50 %) | Approved | 29769116 |
DrugRepV_6627 | Bictegravir | Antiinfectives For Systemic Use | Acquired immunodeficiency syndrome | Human immunodeficiency virus | H51Y (DTG) | | Single-round viral replication assay | Decrease (50 %) | Approved | 29769116 |
DrugRepV_6628 | Bictegravir | Antiinfectives For Systemic Use | Acquired immunodeficiency syndrome | Human immunodeficiency virus | G118R (DTG) | | Single-round viral replication assay | Decrease (50 %) | Approved | 29769116 |
DrugRepV_6629 | Bictegravir | Antiinfectives For Systemic Use | Acquired immunodeficiency syndrome | Human immunodeficiency virus | R263K (DTG) | | Single-round viral replication assay | Decrease (50 %) | Approved | 29769116 |
DrugRepV_6630 | Bictegravir | Antiinfectives For Systemic Use | Acquired immunodeficiency syndrome | Human immunodeficiency virus | H51Y/R263K (DTG) | | Single-round viral replication assay | Decrease (50 %) | Approved | 29769116 |
DrugRepV_6631 | Bictegravir | Antiinfectives For Systemic Use | Acquired immunodeficiency syndrome | Human immunodeficiency virus | E138K/R263K (DTG) | | Single-round viral replication assay | Decrease (50 %) | Approved | 29769116 |
DrugRepV_6632 | Raltegravir | Antiinfectives For Systemic Use | Acquired immunodeficiency syndrome | Human immunodeficiency virus | M50I | | Single-round viral replication assay | Decrease (50 %) | Approved | 29769116 |
DrugRepV_6633 | Raltegravir | Antiinfectives For Systemic Use | Acquired immunodeficiency syndrome | Human immunodeficiency virus | L74M | | Single-round viral replication assay | Decrease (50 %) | Approved | 29769116 |
DrugRepV_6634 | Raltegravir | Antiinfectives For Systemic Use | Acquired immunodeficiency syndrome | Human immunodeficiency virus | T97A | | Single-round viral replication assay | Decrease (50 %) | Approved | 29769116 |
DrugRepV_6635 | Raltegravir | Antiinfectives For Systemic Use | Acquired immunodeficiency syndrome | Human immunodeficiency virus | S119R | | Single-round viral replication assay | Decrease (50 %) | Approved | 29769116 |
DrugRepV_6636 | Raltegravir | Antiinfectives For Systemic Use | Acquired immunodeficiency syndrome | Human immunodeficiency virus | E138K | | Single-round viral replication assay | Decrease (50 %) | Approved | 29769116 |
DrugRepV_6637 | Raltegravir | Antiinfectives For Systemic Use | Acquired immunodeficiency syndrome | Human immunodeficiency virus | G140S | | Single-round viral replication assay | Decrease (50 %) | Approved | 29769116 |
DrugRepV_6638 | Raltegravir | Antiinfectives For Systemic Use | Acquired immunodeficiency syndrome | Human immunodeficiency virus | Q146L | | Single-round viral replication assay | Decrease (50 %) | Approved | 29769116 |
DrugRepV_6639 | Raltegravir | Antiinfectives For Systemic Use | Acquired immunodeficiency syndrome | Human immunodeficiency virus | Q146P | | Single-round viral replication assay | Decrease (50 %) | Approved | 29769116 |
DrugRepV_6640 | Raltegravir | Antiinfectives For Systemic Use | Acquired immunodeficiency syndrome | Human immunodeficiency virus | Q148H | | Single-round viral replication assay | Decrease (50 %) | Approved | 29769116 |
DrugRepV_6641 | Raltegravir | Antiinfectives For Systemic Use | Acquired immunodeficiency syndrome | Human immunodeficiency virus | Q148K | | Single-round viral replication assay | Decrease (50 %) | Approved | 29769116 |
DrugRepV_6642 | Raltegravir | Antiinfectives For Systemic Use | Acquired immunodeficiency syndrome | Human immunodeficiency virus | Q148R | | Single-round viral replication assay | Decrease (50 %) | Approved | 29769116 |
DrugRepV_6643 | Raltegravir | Antiinfectives For Systemic Use | Acquired immunodeficiency syndrome | Human immunodeficiency virus | S153Y | | Single-round viral replication assay | Decrease (50 %) | Approved | 29769116 |
DrugRepV_6644 | Elvitegravir | Antiinfectives For Systemic Use | Acquired immunodeficiency syndrome | Human immunodeficiency virus | M50I | | Single-round viral replication assay | Decrease (50 %) | Approved | 29769116 |
DrugRepV_6645 | Elvitegravir | Antiinfectives For Systemic Use | Acquired immunodeficiency syndrome | Human immunodeficiency virus | L74M | | Single-round viral replication assay | Decrease (50 %) | Approved | 29769116 |
DrugRepV_6646 | Elvitegravir | Antiinfectives For Systemic Use | Acquired immunodeficiency syndrome | Human immunodeficiency virus | T97A | | Single-round viral replication assay | Decrease (50 %) | Approved | 29769116 |
DrugRepV_6647 | Elvitegravir | Antiinfectives For Systemic Use | Acquired immunodeficiency syndrome | Human immunodeficiency virus | S119R | | Single-round viral replication assay | Decrease (50 %) | Approved | 29769116 |
DrugRepV_6648 | Elvitegravir | Antiinfectives For Systemic Use | Acquired immunodeficiency syndrome | Human immunodeficiency virus | E138K | | Single-round viral replication assay | Decrease (50 %) | Approved | 29769116 |
DrugRepV_6649 | Elvitegravir | Antiinfectives For Systemic Use | Acquired immunodeficiency syndrome | Human immunodeficiency virus | G140S | | Single-round viral replication assay | Decrease (50 %) | Approved | 29769116 |
DrugRepV_6650 | Elvitegravir | Antiinfectives For Systemic Use | Acquired immunodeficiency syndrome | Human immunodeficiency virus | Q146L | | Single-round viral replication assay | Decrease (50 %) | Approved | 29769116 |
DrugRepV_6651 | Elvitegravir | Antiinfectives For Systemic Use | Acquired immunodeficiency syndrome | Human immunodeficiency virus | Q146P | | Single-round viral replication assay | Decrease (50 %) | Approved | 29769116 |
DrugRepV_6652 | Elvitegravir | Antiinfectives For Systemic Use | Acquired immunodeficiency syndrome | Human immunodeficiency virus | Q148H | | Single-round viral replication assay | Decrease (50 %) | Approved | 29769116 |
DrugRepV_6653 | Elvitegravir | Antiinfectives For Systemic Use | Acquired immunodeficiency syndrome | Human immunodeficiency virus | Q148K | | Single-round viral replication assay | Decrease (50 %) | Approved | 29769116 |
DrugRepV_6654 | Elvitegravir | Antiinfectives For Systemic Use | Acquired immunodeficiency syndrome | Human immunodeficiency virus | Q148R | | Single-round viral replication assay | Decrease (50 %) | Approved | 29769116 |
DrugRepV_6655 | Elvitegravir | Antiinfectives For Systemic Use | Acquired immunodeficiency syndrome | Human immunodeficiency virus | S153Y | | Single-round viral replication assay | Decrease (50 %) | Approved | 29769116 |
DrugRepV_6656 | Dolutegravir | Antiinfectives For Systemic Use | Acquired immunodeficiency syndrome | Human immunodeficiency virus | M50I | | Single-round viral replication assay | Decrease (50 %) | Approved | 29769116 |
DrugRepV_6657 | Dolutegravir | Antiinfectives For Systemic Use | Acquired immunodeficiency syndrome | Human immunodeficiency virus | L74M | | Single-round viral replication assay | Decrease (50 %) | Approved | 29769116 |
DrugRepV_6658 | Dolutegravir | Antiinfectives For Systemic Use | Acquired immunodeficiency syndrome | Human immunodeficiency virus | T97A | | Single-round viral replication assay | Decrease (50 %) | Approved | 29769116 |
DrugRepV_6659 | Dolutegravir | Antiinfectives For Systemic Use | Acquired immunodeficiency syndrome | Human immunodeficiency virus | S119R | | Single-round viral replication assay | Decrease (50 %) | Approved | 29769116 |
DrugRepV_6660 | Dolutegravir | Antiinfectives For Systemic Use | Acquired immunodeficiency syndrome | Human immunodeficiency virus | E138K | | Single-round viral replication assay | Decrease (50 %) | Approved | 29769116 |
DrugRepV_6661 | Dolutegravir | Antiinfectives For Systemic Use | Acquired immunodeficiency syndrome | Human immunodeficiency virus | G140S | | Single-round viral replication assay | Decrease (50 %) | Approved | 29769116 |
DrugRepV_6662 | Dolutegravir | Antiinfectives For Systemic Use | Acquired immunodeficiency syndrome | Human immunodeficiency virus | Q146L | | Single-round viral replication assay | Decrease (50 %) | Approved | 29769116 |
DrugRepV_6663 | Dolutegravir | Antiinfectives For Systemic Use | Acquired immunodeficiency syndrome | Human immunodeficiency virus | Q146P | | Single-round viral replication assay | Decrease (50 %) | Approved | 29769116 |
DrugRepV_6664 | Dolutegravir | Antiinfectives For Systemic Use | Acquired immunodeficiency syndrome | Human immunodeficiency virus | Q148H | | Single-round viral replication assay | Decrease (50 %) | Approved | 29769116 |
DrugRepV_6665 | Dolutegravir | Antiinfectives For Systemic Use | Acquired immunodeficiency syndrome | Human immunodeficiency virus | Q148K | | Single-round viral replication assay | Decrease (50 %) | Approved | 29769116 |
DrugRepV_6666 | Dolutegravir | Antiinfectives For Systemic Use | Acquired immunodeficiency syndrome | Human immunodeficiency virus | Q148R | | Single-round viral replication assay | Decrease (50 %) | Approved | 29769116 |
DrugRepV_6667 | Dolutegravir | Antiinfectives For Systemic Use | Acquired immunodeficiency syndrome | Human immunodeficiency virus | S153Y | | Single-round viral replication assay | Decrease (50 %) | Approved | 29769116 |
DrugRepV_6668 | Cabotegravir | Antiviral | Acquired immunodeficiency syndrome | Human immunodeficiency virus | M50I | | Single-round viral replication assay | Decrease (50 %) | Phase I | 29769116 |
DrugRepV_6669 | Cabotegravir | Antiviral | Acquired immunodeficiency syndrome | Human immunodeficiency virus | L74M | | Single-round viral replication assay | Decrease (50 %) | Phase I | 29769116 |
DrugRepV_6670 | Cabotegravir | Antiviral | Acquired immunodeficiency syndrome | Human immunodeficiency virus | T97A | | Single-round viral replication assay | Decrease (50 %) | Phase I | 29769116 |
DrugRepV_6671 | Cabotegravir | Antiviral | Acquired immunodeficiency syndrome | Human immunodeficiency virus | S119R | | Single-round viral replication assay | Decrease (50 %) | Phase I | 29769116 |
DrugRepV_6672 | Cabotegravir | Antiviral | Acquired immunodeficiency syndrome | Human immunodeficiency virus | E138K | | Single-round viral replication assay | Decrease (50 %) | Phase I | 29769116 |
DrugRepV_6673 | Cabotegravir | Antiviral | Acquired immunodeficiency syndrome | Human immunodeficiency virus | G140S | | Single-round viral replication assay | Decrease (50 %) | Phase I | 29769116 |
DrugRepV_6674 | Cabotegravir | Antiviral | Acquired immunodeficiency syndrome | Human immunodeficiency virus | Q146L | | Single-round viral replication assay | Decrease (50 %) | Phase I | 29769116 |
DrugRepV_6675 | Cabotegravir | Antiviral | Acquired immunodeficiency syndrome | Human immunodeficiency virus | Q146P | | Single-round viral replication assay | Decrease (50 %) | Phase I | 29769116 |
DrugRepV_6676 | Cabotegravir | Antiviral | Acquired immunodeficiency syndrome | Human immunodeficiency virus | Q148H | | Single-round viral replication assay | Decrease (50 %) | Phase I | 29769116 |
DrugRepV_6677 | Cabotegravir | Antiviral | Acquired immunodeficiency syndrome | Human immunodeficiency virus | Q148K | | Single-round viral replication assay | Decrease (50 %) | Phase I | 29769116 |
DrugRepV_6678 | Cabotegravir | Antiviral | Acquired immunodeficiency syndrome | Human immunodeficiency virus | Q148R | | Single-round viral replication assay | Decrease (50 %) | Phase I | 29769116 |
DrugRepV_6679 | Cabotegravir | Antiviral | Acquired immunodeficiency syndrome | Human immunodeficiency virus | S153Y | | Single-round viral replication assay | Decrease (50 %) | Phase I | 29769116 |
DrugRepV_6680 | Bictegravir | Antiinfectives For Systemic Use | Acquired immunodeficiency syndrome | Human immunodeficiency virus | M50I | | Single-round viral replication assay | Decrease (50 %) | Approved | 29769116 |
DrugRepV_6681 | Bictegravir | Antiinfectives For Systemic Use | Acquired immunodeficiency syndrome | Human immunodeficiency virus | L74M | | Single-round viral replication assay | Decrease (50 %) | Approved | 29769116 |
DrugRepV_6682 | Bictegravir | Antiinfectives For Systemic Use | Acquired immunodeficiency syndrome | Human immunodeficiency virus | T97A | | Single-round viral replication assay | Decrease (50 %) | Approved | 29769116 |
DrugRepV_6683 | Bictegravir | Antiinfectives For Systemic Use | Acquired immunodeficiency syndrome | Human immunodeficiency virus | S119R | | Single-round viral replication assay | Decrease (50 %) | Approved | 29769116 |
DrugRepV_6684 | Bictegravir | Antiinfectives For Systemic Use | Acquired immunodeficiency syndrome | Human immunodeficiency virus | E138K | | Single-round viral replication assay | Decrease (50 %) | Approved | 29769116 |
DrugRepV_6685 | Bictegravir | Antiinfectives For Systemic Use | Acquired immunodeficiency syndrome | Human immunodeficiency virus | G140S | | Single-round viral replication assay | Decrease (50 %) | Approved | 29769116 |
DrugRepV_6686 | Bictegravir | Antiinfectives For Systemic Use | Acquired immunodeficiency syndrome | Human immunodeficiency virus | Q146L | | Single-round viral replication assay | Decrease (50 %) | Approved | 29769116 |
DrugRepV_6687 | Bictegravir | Antiinfectives For Systemic Use | Acquired immunodeficiency syndrome | Human immunodeficiency virus | Q146P | | Single-round viral replication assay | Decrease (50 %) | Approved | 29769116 |
DrugRepV_6688 | Bictegravir | Antiinfectives For Systemic Use | Acquired immunodeficiency syndrome | Human immunodeficiency virus | Q148H | | Single-round viral replication assay | Decrease (50 %) | Approved | 29769116 |
DrugRepV_6689 | Bictegravir | Antiinfectives For Systemic Use | Acquired immunodeficiency syndrome | Human immunodeficiency virus | Q148K | | Single-round viral replication assay | Decrease (50 %) | Approved | 29769116 |
DrugRepV_6690 | Bictegravir | Antiinfectives For Systemic Use | Acquired immunodeficiency syndrome | Human immunodeficiency virus | Q148R | | Single-round viral replication assay | Decrease (50 %) | Approved | 29769116 |
DrugRepV_6691 | Bictegravir | Antiinfectives For Systemic Use | Acquired immunodeficiency syndrome | Human immunodeficiency virus | S153Y | | Single-round viral replication assay | Decrease (50 %) | Approved | 29769116 |
DrugRepV_6692 | Raltegravir | Antiinfectives For Systemic Use | Acquired immunodeficiency syndrome | Human immunodeficiency virus | G140A/Q148H | | Single-round viral replication assay | Decrease (50 %) | Approved | 29769116 |
DrugRepV_6693 | Raltegravir | Antiinfectives For Systemic Use | Acquired immunodeficiency syndrome | Human immunodeficiency virus | Y143R/Q148H | | Single-round viral replication assay | Decrease (50 %) | Approved | 29769116 |
DrugRepV_6694 | Raltegravir | Antiinfectives For Systemic Use | Acquired immunodeficiency syndrome | Human immunodeficiency virus | Q148H/N155H | | Single-round viral replication assay | Decrease (50 %) | Approved | 29769116 |
DrugRepV_6695 | Raltegravir | Antiinfectives For Systemic Use | Acquired immunodeficiency syndrome | Human immunodeficiency virus | E138K/Q148K | | Single-round viral replication assay | Decrease (50 %) | Approved | 29769116 |
DrugRepV_6696 | Raltegravir | Antiinfectives For Systemic Use | Acquired immunodeficiency syndrome | Human immunodeficiency virus | G140A/Q148K | | Single-round viral replication assay | Decrease (50 %) | Approved | 29769116 |
DrugRepV_6697 | Raltegravir | Antiinfectives For Systemic Use | Acquired immunodeficiency syndrome | Human immunodeficiency virus | G140S/Q148K | | Single-round viral replication assay | Decrease (50 %) | Approved | 29769116 |
DrugRepV_6698 | Raltegravir | Antiinfectives For Systemic Use | Acquired immunodeficiency syndrome | Human immunodeficiency virus | E138A/Q148R | | Single-round viral replication assay | Decrease (50 %) | Approved | 29769116 |
DrugRepV_6699 | Raltegravir | Antiinfectives For Systemic Use | Acquired immunodeficiency syndrome | Human immunodeficiency virus | E138K/Q148R | | Single-round viral replication assay | Decrease (50 %) | Approved | 29769116 |
DrugRepV_6700 | Raltegravir | Antiinfectives For Systemic Use | Acquired immunodeficiency syndrome | Human immunodeficiency virus | G140A/Q148R | | Single-round viral replication assay | Decrease (50 %) | Approved | 29769116 |
DrugRepV_6701 | Raltegravir | Antiinfectives For Systemic Use | Acquired immunodeficiency syndrome | Human immunodeficiency virus | G140C/Q148R | | Single-round viral replication assay | Decrease (50 %) | Approved | 29769116 |
DrugRepV_6702 | Raltegravir | Antiinfectives For Systemic Use | Acquired immunodeficiency syndrome | Human immunodeficiency virus | G140S/Q148R | | Single-round viral replication assay | Decrease (50 %) | Approved | 29769116 |
DrugRepV_6703 | Raltegravir | Antiinfectives For Systemic Use | Acquired immunodeficiency syndrome | Human immunodeficiency virus | Q148R/N155H | | Single-round viral replication assay | Decrease (50 %) | Approved | 29769116 |
DrugRepV_6704 | Elvitegravir | Antiinfectives For Systemic Use | Acquired immunodeficiency syndrome | Human immunodeficiency virus | G140A/Q148H | | Single-round viral replication assay | Decrease (50 %) | Approved | 29769116 |
DrugRepV_6705 | Elvitegravir | Antiinfectives For Systemic Use | Acquired immunodeficiency syndrome | Human immunodeficiency virus | Y143R/Q148H | | Single-round viral replication assay | Decrease (50 %) | Approved | 29769116 |
DrugRepV_6706 | Elvitegravir | Antiinfectives For Systemic Use | Acquired immunodeficiency syndrome | Human immunodeficiency virus | Q148H/N155H | | Single-round viral replication assay | Decrease (50 %) | Approved | 29769116 |
DrugRepV_6707 | Elvitegravir | Antiinfectives For Systemic Use | Acquired immunodeficiency syndrome | Human immunodeficiency virus | E138K/Q148K | | Single-round viral replication assay | Decrease (50 %) | Approved | 29769116 |
DrugRepV_6708 | Elvitegravir | Antiinfectives For Systemic Use | Acquired immunodeficiency syndrome | Human immunodeficiency virus | G140A/Q148K | | Single-round viral replication assay | Decrease (50 %) | Approved | 29769116 |
DrugRepV_6709 | Elvitegravir | Antiinfectives For Systemic Use | Acquired immunodeficiency syndrome | Human immunodeficiency virus | G140S/Q148K | | Single-round viral replication assay | Decrease (50 %) | Approved | 29769116 |
DrugRepV_6710 | Elvitegravir | Antiinfectives For Systemic Use | Acquired immunodeficiency syndrome | Human immunodeficiency virus | E138A/Q148R | | Single-round viral replication assay | Decrease (50 %) | Approved | 29769116 |
DrugRepV_6711 | Elvitegravir | Antiinfectives For Systemic Use | Acquired immunodeficiency syndrome | Human immunodeficiency virus | E138K/Q148R | | Single-round viral replication assay | Decrease (50 %) | Approved | 29769116 |
DrugRepV_6712 | Elvitegravir | Antiinfectives For Systemic Use | Acquired immunodeficiency syndrome | Human immunodeficiency virus | G140A/Q148R | | Single-round viral replication assay | Decrease (50 %) | Approved | 29769116 |
DrugRepV_6713 | Elvitegravir | Antiinfectives For Systemic Use | Acquired immunodeficiency syndrome | Human immunodeficiency virus | G140C/Q148R | | Single-round viral replication assay | Decrease (50 %) | Approved | 29769116 |
DrugRepV_6714 | Elvitegravir | Antiinfectives For Systemic Use | Acquired immunodeficiency syndrome | Human immunodeficiency virus | G140S/Q148R | | Single-round viral replication assay | Decrease (50 %) | Approved | 29769116 |
DrugRepV_6715 | Elvitegravir | Antiinfectives For Systemic Use | Acquired immunodeficiency syndrome | Human immunodeficiency virus | Q148R/N155H | | Single-round viral replication assay | Decrease (50 %) | Approved | 29769116 |
DrugRepV_6716 | Dolutegravir | Antiinfectives For Systemic Use | Acquired immunodeficiency syndrome | Human immunodeficiency virus | G140A/Q148H | | Single-round viral replication assay | Decrease (50 %) | Approved | 29769116 |
DrugRepV_6717 | Dolutegravir | Antiinfectives For Systemic Use | Acquired immunodeficiency syndrome | Human immunodeficiency virus | Y143R/Q148H | | Single-round viral replication assay | Decrease (50 %) | Approved | 29769116 |
DrugRepV_6718 | Dolutegravir | Antiinfectives For Systemic Use | Acquired immunodeficiency syndrome | Human immunodeficiency virus | Q148H/N155H | | Single-round viral replication assay | Decrease (50 %) | Approved | 29769116 |
DrugRepV_6719 | Dolutegravir | Antiinfectives For Systemic Use | Acquired immunodeficiency syndrome | Human immunodeficiency virus | E138K/Q148K | | Single-round viral replication assay | Decrease (50 %) | Approved | 29769116 |
DrugRepV_6720 | Dolutegravir | Antiinfectives For Systemic Use | Acquired immunodeficiency syndrome | Human immunodeficiency virus | G140A/Q148K | | Single-round viral replication assay | Decrease (50 %) | Approved | 29769116 |
DrugRepV_6721 | Dolutegravir | Antiinfectives For Systemic Use | Acquired immunodeficiency syndrome | Human immunodeficiency virus | G140S/Q148K | | Single-round viral replication assay | Decrease (50 %) | Approved | 29769116 |
DrugRepV_6722 | Dolutegravir | Antiinfectives For Systemic Use | Acquired immunodeficiency syndrome | Human immunodeficiency virus | E138A/Q148R | | Single-round viral replication assay | Decrease (50 %) | Approved | 29769116 |
DrugRepV_6723 | Dolutegravir | Antiinfectives For Systemic Use | Acquired immunodeficiency syndrome | Human immunodeficiency virus | E138K/Q148R | | Single-round viral replication assay | Decrease (50 %) | Approved | 29769116 |
DrugRepV_6724 | Dolutegravir | Antiinfectives For Systemic Use | Acquired immunodeficiency syndrome | Human immunodeficiency virus | G140A/Q148R | | Single-round viral replication assay | Decrease (50 %) | Approved | 29769116 |
DrugRepV_6725 | Dolutegravir | Antiinfectives For Systemic Use | Acquired immunodeficiency syndrome | Human immunodeficiency virus | G140C/Q148R | | Single-round viral replication assay | Decrease (50 %) | Approved | 29769116 |
DrugRepV_6726 | Dolutegravir | Antiinfectives For Systemic Use | Acquired immunodeficiency syndrome | Human immunodeficiency virus | G140S/Q148R | | Single-round viral replication assay | Decrease (50 %) | Approved | 29769116 |
DrugRepV_6727 | Dolutegravir | Antiinfectives For Systemic Use | Acquired immunodeficiency syndrome | Human immunodeficiency virus | Q148R/N155H | | Single-round viral replication assay | Decrease (50 %) | Approved | 29769116 |
DrugRepV_6728 | Cabotegravir | Antiviral | Acquired immunodeficiency syndrome | Human immunodeficiency virus | G140A/Q148H | | Single-round viral replication assay | Decrease (50 %) | Phase I | 29769116 |
DrugRepV_6729 | Cabotegravir | Antiviral | Acquired immunodeficiency syndrome | Human immunodeficiency virus | Y143R/Q148H | | Single-round viral replication assay | Decrease (50 %) | Phase I | 29769116 |
DrugRepV_6730 | Cabotegravir | Antiviral | Acquired immunodeficiency syndrome | Human immunodeficiency virus | Q148H/N155H | | Single-round viral replication assay | Decrease (50 %) | Phase I | 29769116 |
DrugRepV_6731 | Cabotegravir | Antiviral | Acquired immunodeficiency syndrome | Human immunodeficiency virus | E138K/Q148K | | Single-round viral replication assay | Decrease (50 %) | Phase I | 29769116 |
DrugRepV_6732 | Cabotegravir | Antiviral | Acquired immunodeficiency syndrome | Human immunodeficiency virus | G140A/Q148K | | Single-round viral replication assay | Decrease (50 %) | Phase I | 29769116 |
DrugRepV_6733 | Cabotegravir | Antiviral | Acquired immunodeficiency syndrome | Human immunodeficiency virus | G140S/Q148K | | Single-round viral replication assay | Decrease (50 %) | Phase I | 29769116 |
DrugRepV_6734 | Cabotegravir | Antiviral | Acquired immunodeficiency syndrome | Human immunodeficiency virus | E138A/Q148R | | Single-round viral replication assay | Decrease (50 %) | Phase I | 29769116 |
DrugRepV_6735 | Cabotegravir | Antiviral | Acquired immunodeficiency syndrome | Human immunodeficiency virus | E138K/Q148R | | Single-round viral replication assay | Decrease (50 %) | Phase I | 29769116 |
DrugRepV_6736 | Cabotegravir | Antiviral | Acquired immunodeficiency syndrome | Human immunodeficiency virus | G140A/Q148R | | Single-round viral replication assay | Decrease (50 %) | Phase I | 29769116 |
DrugRepV_6737 | Cabotegravir | Antiviral | Acquired immunodeficiency syndrome | Human immunodeficiency virus | G140C/Q148R | | Single-round viral replication assay | Decrease (50 %) | Phase I | 29769116 |
DrugRepV_6738 | Cabotegravir | Antiviral | Acquired immunodeficiency syndrome | Human immunodeficiency virus | G140S/Q148R | | Single-round viral replication assay | Decrease (50 %) | Phase I | 29769116 |
DrugRepV_6739 | Cabotegravir | Antiviral | Acquired immunodeficiency syndrome | Human immunodeficiency virus | Q148R/N155H | | Single-round viral replication assay | Decrease (50 %) | Phase I | 29769116 |
DrugRepV_6740 | Bictegravir | Antiinfectives For Systemic Use | Acquired immunodeficiency syndrome | Human immunodeficiency virus | G140A/Q148H | | Single-round viral replication assay | Decrease (50 %) | Approved | 29769116 |
DrugRepV_6741 | Bictegravir | Antiinfectives For Systemic Use | Acquired immunodeficiency syndrome | Human immunodeficiency virus | Y143R/Q148H | | Single-round viral replication assay | Decrease (50 %) | Approved | 29769116 |
DrugRepV_6742 | Bictegravir | Antiinfectives For Systemic Use | Acquired immunodeficiency syndrome | Human immunodeficiency virus | Q148H/N155H | | Single-round viral replication assay | Decrease (50 %) | Approved | 29769116 |
DrugRepV_6743 | Bictegravir | Antiinfectives For Systemic Use | Acquired immunodeficiency syndrome | Human immunodeficiency virus | E138K/Q148K | | Single-round viral replication assay | Decrease (50 %) | Approved | 29769116 |
DrugRepV_6744 | Bictegravir | Antiinfectives For Systemic Use | Acquired immunodeficiency syndrome | Human immunodeficiency virus | G140A/Q148K | | Single-round viral replication assay | Decrease (50 %) | Approved | 29769116 |
DrugRepV_6745 | Bictegravir | Antiinfectives For Systemic Use | Acquired immunodeficiency syndrome | Human immunodeficiency virus | G140S/Q148K | | Single-round viral replication assay | Decrease (50 %) | Approved | 29769116 |
DrugRepV_6746 | Bictegravir | Antiinfectives For Systemic Use | Acquired immunodeficiency syndrome | Human immunodeficiency virus | E138A/Q148R | | Single-round viral replication assay | Decrease (50 %) | Approved | 29769116 |
DrugRepV_6747 | Bictegravir | Antiinfectives For Systemic Use | Acquired immunodeficiency syndrome | Human immunodeficiency virus | E138K/Q148R | | Single-round viral replication assay | Decrease (50 %) | Approved | 29769116 |
DrugRepV_6748 | Bictegravir | Antiinfectives For Systemic Use | Acquired immunodeficiency syndrome | Human immunodeficiency virus | G140A/Q148R | | Single-round viral replication assay | Decrease (50 %) | Approved | 29769116 |
DrugRepV_6749 | Bictegravir | Antiinfectives For Systemic Use | Acquired immunodeficiency syndrome | Human immunodeficiency virus | G140C/Q148R | | Single-round viral replication assay | Decrease (50 %) | Approved | 29769116 |
DrugRepV_6750 | Bictegravir | Antiinfectives For Systemic Use | Acquired immunodeficiency syndrome | Human immunodeficiency virus | G140S/Q148R | | Single-round viral replication assay | Decrease (50 %) | Approved | 29769116 |
DrugRepV_6751 | Bictegravir | Antiinfectives For Systemic Use | Acquired immunodeficiency syndrome | Human immunodeficiency virus | Q148R/N155H | | Single-round viral replication assay | Decrease (50 %) | Approved | 29769116 |
DrugRepV_6752 | Raltegravir | Antiinfectives For Systemic Use | Acquired immunodeficiency syndrome | Human immunodeficiency virus | T66I/E157Q | | Single-round viral replication assay | Decrease (50 %) | Approved | 29769116 |
DrugRepV_6753 | Raltegravir | Antiinfectives For Systemic Use | Acquired immunodeficiency syndrome | Human immunodeficiency virus | E92Q/N155H | | Single-round viral replication assay | Decrease (50 %) | Approved | 29769116 |
DrugRepV_6754 | Raltegravir | Antiinfectives For Systemic Use | Acquired immunodeficiency syndrome | Human immunodeficiency virus | G140S/N155H | | Single-round viral replication assay | Decrease (50 %) | Approved | 29769116 |
DrugRepV_6755 | Raltegravir | Antiinfectives For Systemic Use | Acquired immunodeficiency syndrome | Human immunodeficiency virus | Y143H/N155H | | Single-round viral replication assay | Decrease (50 %) | Approved | 29769116 |
DrugRepV_6756 | Raltegravir | Antiinfectives For Systemic Use | Acquired immunodeficiency syndrome | Human immunodeficiency virus | Y143R/N155H | | Single-round viral replication assay | Decrease (50 %) | Approved | 29769116 |
DrugRepV_6757 | Raltegravir | Antiinfectives For Systemic Use | Acquired immunodeficiency syndrome | Human immunodeficiency virus | N155H/G163R | | Single-round viral replication assay | Decrease (50 %) | Approved | 29769116 |
DrugRepV_6758 | Elvitegravir | Antiinfectives For Systemic Use | Acquired immunodeficiency syndrome | Human immunodeficiency virus | T66I/E157Q | | Single-round viral replication assay | Decrease (50 %) | Approved | 29769116 |
DrugRepV_6759 | Elvitegravir | Antiinfectives For Systemic Use | Acquired immunodeficiency syndrome | Human immunodeficiency virus | E92Q/N155H | | Single-round viral replication assay | Decrease (50 %) | Approved | 29769116 |
DrugRepV_6760 | Elvitegravir | Antiinfectives For Systemic Use | Acquired immunodeficiency syndrome | Human immunodeficiency virus | G140S/N155H | | Single-round viral replication assay | Decrease (50 %) | Approved | 29769116 |
DrugRepV_6761 | Elvitegravir | Antiinfectives For Systemic Use | Acquired immunodeficiency syndrome | Human immunodeficiency virus | Y143H/N155H | | Single-round viral replication assay | Decrease (50 %) | Approved | 29769116 |
DrugRepV_6762 | Elvitegravir | Antiinfectives For Systemic Use | Acquired immunodeficiency syndrome | Human immunodeficiency virus | Y143R/N155H | | Single-round viral replication assay | Decrease (50 %) | Approved | 29769116 |
DrugRepV_6763 | Elvitegravir | Antiinfectives For Systemic Use | Acquired immunodeficiency syndrome | Human immunodeficiency virus | N155H/G163R | | Single-round viral replication assay | Decrease (50 %) | Approved | 29769116 |
DrugRepV_6764 | Dolutegravir | Antiinfectives For Systemic Use | Acquired immunodeficiency syndrome | Human immunodeficiency virus | T66I/E157Q | | Single-round viral replication assay | Decrease (50 %) | Approved | 29769116 |
DrugRepV_6765 | Dolutegravir | Antiinfectives For Systemic Use | Acquired immunodeficiency syndrome | Human immunodeficiency virus | E92Q/N155H | | Single-round viral replication assay | Decrease (50 %) | Approved | 29769116 |
DrugRepV_6766 | Dolutegravir | Antiinfectives For Systemic Use | Acquired immunodeficiency syndrome | Human immunodeficiency virus | G140S/N155H | | Single-round viral replication assay | Decrease (50 %) | Approved | 29769116 |
DrugRepV_6767 | Dolutegravir | Antiinfectives For Systemic Use | Acquired immunodeficiency syndrome | Human immunodeficiency virus | Y143H/N155H | | Single-round viral replication assay | Decrease (50 %) | Approved | 29769116 |
DrugRepV_6768 | Dolutegravir | Antiinfectives For Systemic Use | Acquired immunodeficiency syndrome | Human immunodeficiency virus | Y143R/N155H | | Single-round viral replication assay | Decrease (50 %) | Approved | 29769116 |
DrugRepV_6769 | Dolutegravir | Antiinfectives For Systemic Use | Acquired immunodeficiency syndrome | Human immunodeficiency virus | N155H/G163R | | Single-round viral replication assay | Decrease (50 %) | Approved | 29769116 |
DrugRepV_6770 | Cabotegravir | Antiviral | Acquired immunodeficiency syndrome | Human immunodeficiency virus | T66I/E157Q | | Single-round viral replication assay | Decrease (50 %) | Phase I | 29769116 |
DrugRepV_6771 | Cabotegravir | Antiviral | Acquired immunodeficiency syndrome | Human immunodeficiency virus | E92Q/N155H | | Single-round viral replication assay | Decrease (50 %) | Phase I | 29769116 |
DrugRepV_6772 | Cabotegravir | Antiviral | Acquired immunodeficiency syndrome | Human immunodeficiency virus | G140S/N155H | | Single-round viral replication assay | Decrease (50 %) | Phase I | 29769116 |
DrugRepV_6773 | Cabotegravir | Antiviral | Acquired immunodeficiency syndrome | Human immunodeficiency virus | Y143H/N155H | | Single-round viral replication assay | Decrease (50 %) | Phase I | 29769116 |
DrugRepV_6774 | Cabotegravir | Antiviral | Acquired immunodeficiency syndrome | Human immunodeficiency virus | Y143R/N155H | | Single-round viral replication assay | Decrease (50 %) | Phase I | 29769116 |
DrugRepV_6775 | Cabotegravir | Antiviral | Acquired immunodeficiency syndrome | Human immunodeficiency virus | N155H/G163R | | Single-round viral replication assay | Decrease (50 %) | Phase I | 29769116 |
DrugRepV_6776 | Bictegravir | Antiinfectives For Systemic Use | Acquired immunodeficiency syndrome | Human immunodeficiency virus | T66I/E157Q | | Single-round viral replication assay | Decrease (50 %) | Approved | 29769116 |
DrugRepV_6777 | Bictegravir | Antiinfectives For Systemic Use | Acquired immunodeficiency syndrome | Human immunodeficiency virus | E92Q/N155H | | Single-round viral replication assay | Decrease (50 %) | Approved | 29769116 |
DrugRepV_6778 | Bictegravir | Antiinfectives For Systemic Use | Acquired immunodeficiency syndrome | Human immunodeficiency virus | G140S/N155H | | Single-round viral replication assay | Decrease (50 %) | Approved | 29769116 |
DrugRepV_6779 | Bictegravir | Antiinfectives For Systemic Use | Acquired immunodeficiency syndrome | Human immunodeficiency virus | Y143H/N155H | | Single-round viral replication assay | Decrease (50 %) | Approved | 29769116 |
DrugRepV_6780 | Bictegravir | Antiinfectives For Systemic Use | Acquired immunodeficiency syndrome | Human immunodeficiency virus | Y143R/N155H | | Single-round viral replication assay | Decrease (50 %) | Approved | 29769116 |
DrugRepV_6781 | Bictegravir | Antiinfectives For Systemic Use | Acquired immunodeficiency syndrome | Human immunodeficiency virus | N155H/G163R | | Single-round viral replication assay | Decrease (50 %) | Approved | 29769116 |
DrugRepV_6782 | Raltegravir | Antiinfectives For Systemic Use | Acquired immunodeficiency syndrome | Human immunodeficiency virus | 97A/Y143R/Q148H | | Single-round viral replication assay | Decrease (50 %) | Approved | 29769116 |
DrugRepV_6783 | Raltegravir | Antiinfectives For Systemic Use | Acquired immunodeficiency syndrome | Human immunodeficiency virus | T97A/Q148H/N155H | | Single-round viral replication assay | Decrease (50 %) | Approved | 29769116 |
DrugRepV_6784 | Raltegravir | Antiinfectives For Systemic Use | Acquired immunodeficiency syndrome | Human immunodeficiency virus | E138K/G140A/Q148K | | Single-round viral replication assay | Decrease (50 %) | Approved | 29769116 |
DrugRepV_6785 | Raltegravir | Antiinfectives For Systemic Use | Acquired immunodeficiency syndrome | Human immunodeficiency virus | L74M/G140A/Q148R | | Single-round viral replication assay | Decrease (50 %) | Approved | 29769116 |
DrugRepV_6786 | Raltegravir | Antiinfectives For Systemic Use | Acquired immunodeficiency syndrome | Human immunodeficiency virus | L74M/G140C/Q148R | | Single-round viral replication assay | Decrease (50 %) | Approved | 29769116 |
DrugRepV_6787 | Raltegravir | Antiinfectives For Systemic Use | Acquired immunodeficiency syndrome | Human immunodeficiency virus | E138K/G140C/Q148R | | Single-round viral replication assay | Decrease (50 %) | Approved | 29769116 |
DrugRepV_6788 | Raltegravir | Antiinfectives For Systemic Use | Acquired immunodeficiency syndrome | Human immunodeficiency virus | E138A/S147G/Q148R | | Single-round viral replication assay | Decrease (50 %) | Approved | 29769116 |
DrugRepV_6789 | Elvitegravir | Antiinfectives For Systemic Use | Acquired immunodeficiency syndrome | Human immunodeficiency virus | 97A/Y143R/Q148H | | Single-round viral replication assay | Decrease (50 %) | Approved | 29769116 |
DrugRepV_6790 | Elvitegravir | Antiinfectives For Systemic Use | Acquired immunodeficiency syndrome | Human immunodeficiency virus | T97A/Q148H/N155H | | Single-round viral replication assay | Decrease (50 %) | Approved | 29769116 |
DrugRepV_6791 | Elvitegravir | Antiinfectives For Systemic Use | Acquired immunodeficiency syndrome | Human immunodeficiency virus | E138K/G140A/Q148K | | Single-round viral replication assay | Decrease (50 %) | Approved | 29769116 |
DrugRepV_6792 | Elvitegravir | Antiinfectives For Systemic Use | Acquired immunodeficiency syndrome | Human immunodeficiency virus | L74M/G140A/Q148R | | Single-round viral replication assay | Decrease (50 %) | Approved | 29769116 |
DrugRepV_6793 | Elvitegravir | Antiinfectives For Systemic Use | Acquired immunodeficiency syndrome | Human immunodeficiency virus | L74M/G140C/Q148R | | Single-round viral replication assay | Decrease (50 %) | Approved | 29769116 |
DrugRepV_6794 | Elvitegravir | Antiinfectives For Systemic Use | Acquired immunodeficiency syndrome | Human immunodeficiency virus | E138K/G140C/Q148R | | Single-round viral replication assay | Decrease (50 %) | Approved | 29769116 |
DrugRepV_6795 | Elvitegravir | Antiinfectives For Systemic Use | Acquired immunodeficiency syndrome | Human immunodeficiency virus | E138A/S147G/Q148R | | Single-round viral replication assay | Decrease (50 %) | Approved | 29769116 |
DrugRepV_6796 | Dolutegravir | Antiinfectives For Systemic Use | Acquired immunodeficiency syndrome | Human immunodeficiency virus | 97A/Y143R/Q148H | | Single-round viral replication assay | Decrease (50 %) | Approved | 29769116 |
DrugRepV_6797 | Dolutegravir | Antiinfectives For Systemic Use | Acquired immunodeficiency syndrome | Human immunodeficiency virus | T97A/Q148H/N155H | | Single-round viral replication assay | Decrease (50 %) | Approved | 29769116 |
DrugRepV_6798 | Dolutegravir | Antiinfectives For Systemic Use | Acquired immunodeficiency syndrome | Human immunodeficiency virus | E138K/G140A/Q148K | | Single-round viral replication assay | Decrease (50 %) | Approved | 29769116 |
DrugRepV_6799 | Dolutegravir | Antiinfectives For Systemic Use | Acquired immunodeficiency syndrome | Human immunodeficiency virus | L74M/G140A/Q148R | | Single-round viral replication assay | Decrease (50 %) | Approved | 29769116 |
DrugRepV_6800 | Dolutegravir | Antiinfectives For Systemic Use | Acquired immunodeficiency syndrome | Human immunodeficiency virus | L74M/G140C/Q148R | | Single-round viral replication assay | Decrease (50 %) | Approved | 29769116 |
DrugRepV_6801 | Dolutegravir | Antiinfectives For Systemic Use | Acquired immunodeficiency syndrome | Human immunodeficiency virus | E138K/G140C/Q148R | | Single-round viral replication assay | Decrease (50 %) | Approved | 29769116 |
DrugRepV_6802 | Dolutegravir | Antiinfectives For Systemic Use | Acquired immunodeficiency syndrome | Human immunodeficiency virus | E138A/S147G/Q148R | | Single-round viral replication assay | Decrease (50 %) | Approved | 29769116 |
DrugRepV_6803 | Cabotegravir | Antiviral | Acquired immunodeficiency syndrome | Human immunodeficiency virus | 97A/Y143R/Q148H | | Single-round viral replication assay | Decrease (50 %) | Phase I | 29769116 |
DrugRepV_6804 | Cabotegravir | Antiviral | Acquired immunodeficiency syndrome | Human immunodeficiency virus | T97A/Q148H/N155H | | Single-round viral replication assay | Decrease (50 %) | Phase I | 29769116 |
DrugRepV_6805 | Cabotegravir | Antiviral | Acquired immunodeficiency syndrome | Human immunodeficiency virus | E138K/G140A/Q148K | | Single-round viral replication assay | Decrease (50 %) | Phase I | 29769116 |
DrugRepV_6806 | Cabotegravir | Antiviral | Acquired immunodeficiency syndrome | Human immunodeficiency virus | L74M/G140A/Q148R | | Single-round viral replication assay | Decrease (50 %) | Phase I | 29769116 |
DrugRepV_6807 | Cabotegravir | Antiviral | Acquired immunodeficiency syndrome | Human immunodeficiency virus | L74M/G140C/Q148R | | Single-round viral replication assay | Decrease (50 %) | Phase I | 29769116 |
DrugRepV_6808 | Cabotegravir | Antiviral | Acquired immunodeficiency syndrome | Human immunodeficiency virus | E138K/G140C/Q148R | | Single-round viral replication assay | Decrease (50 %) | Phase I | 29769116 |
DrugRepV_6809 | Cabotegravir | Antiviral | Acquired immunodeficiency syndrome | Human immunodeficiency virus | E138A/S147G/Q148R | | Single-round viral replication assay | Decrease (50 %) | Phase I | 29769116 |
DrugRepV_6810 | Bictegravir | Antiinfectives For Systemic Use | Acquired immunodeficiency syndrome | Human immunodeficiency virus | 97A/Y143R/Q148H | | Single-round viral replication assay | Decrease (50 %) | Approved | 29769116 |
DrugRepV_6811 | Bictegravir | Antiinfectives For Systemic Use | Acquired immunodeficiency syndrome | Human immunodeficiency virus | T97A/Q148H/N155H | | Single-round viral replication assay | Decrease (50 %) | Approved | 29769116 |
DrugRepV_6812 | Bictegravir | Antiinfectives For Systemic Use | Acquired immunodeficiency syndrome | Human immunodeficiency virus | E138K/G140A/Q148K | | Single-round viral replication assay | Decrease (50 %) | Approved | 29769116 |
DrugRepV_6813 | Bictegravir | Antiinfectives For Systemic Use | Acquired immunodeficiency syndrome | Human immunodeficiency virus | L74M/G140A/Q148R | | Single-round viral replication assay | Decrease (50 %) | Approved | 29769116 |
DrugRepV_6814 | Bictegravir | Antiinfectives For Systemic Use | Acquired immunodeficiency syndrome | Human immunodeficiency virus | L74M/G140C/Q148R | | Single-round viral replication assay | Decrease (50 %) | Approved | 29769116 |
DrugRepV_6815 | Bictegravir | Antiinfectives For Systemic Use | Acquired immunodeficiency syndrome | Human immunodeficiency virus | E138K/G140C/Q148R | | Single-round viral replication assay | Decrease (50 %) | Approved | 29769116 |
DrugRepV_6816 | Bictegravir | Antiinfectives For Systemic Use | Acquired immunodeficiency syndrome | Human immunodeficiency virus | E138A/S147G/Q148R | | Single-round viral replication assay | Decrease (50 %) | Approved | 29769116 |
DrugRepV_6817 | Raltegravir | Antiinfectives For Systemic Use | Acquired immunodeficiency syndrome | Human immunodeficiency virus | T66I/T97A/E157Q | | Single-round viral replication assay | Decrease (50 %) | Approved | 29769116 |
DrugRepV_6818 | Raltegravir | Antiinfectives For Systemic Use | Acquired immunodeficiency syndrome | Human immunodeficiency virus | T97A/Y143R/N155H | | Single-round viral replication assay | Decrease (50 %) | Approved | 29769116 |
DrugRepV_6819 | Raltegravir | Antiinfectives For Systemic Use | Acquired immunodeficiency syndrome | Human immunodeficiency virus | G140S/Y143R/N155H | | Single-round viral replication assay | Decrease (50 %) | Approved | 29769116 |
DrugRepV_6820 | Raltegravir | Antiinfectives For Systemic Use | Acquired immunodeficiency syndrome | Human immunodeficiency virus | E92Q/N155H/G163R | | Single-round viral replication assay | Decrease (50 %) | Approved | 29769116 |
DrugRepV_6821 | Elvitegravir | Antiinfectives For Systemic Use | Acquired immunodeficiency syndrome | Human immunodeficiency virus | T66I/T97A/E157Q | | Single-round viral replication assay | Decrease (50 %) | Approved | 29769116 |
DrugRepV_6822 | Elvitegravir | Antiinfectives For Systemic Use | Acquired immunodeficiency syndrome | Human immunodeficiency virus | T97A/Y143R/N155H | | Single-round viral replication assay | Decrease (50 %) | Approved | 29769116 |
DrugRepV_6823 | Elvitegravir | Antiinfectives For Systemic Use | Acquired immunodeficiency syndrome | Human immunodeficiency virus | G140S/Y143R/N155H | | Single-round viral replication assay | Decrease (50 %) | Approved | 29769116 |
DrugRepV_6824 | Elvitegravir | Antiinfectives For Systemic Use | Acquired immunodeficiency syndrome | Human immunodeficiency virus | E92Q/N155H/G163R | | Single-round viral replication assay | Decrease (50 %) | Approved | 29769116 |
DrugRepV_6825 | Dolutegravir | Antiinfectives For Systemic Use | Acquired immunodeficiency syndrome | Human immunodeficiency virus | T66I/T97A/E157Q | | Single-round viral replication assay | Decrease (50 %) | Approved | 29769116 |
DrugRepV_6826 | Dolutegravir | Antiinfectives For Systemic Use | Acquired immunodeficiency syndrome | Human immunodeficiency virus | T97A/Y143R/N155H | | Single-round viral replication assay | Decrease (50 %) | Approved | 29769116 |
DrugRepV_6827 | Dolutegravir | Antiinfectives For Systemic Use | Acquired immunodeficiency syndrome | Human immunodeficiency virus | G140S/Y143R/N155H | | Single-round viral replication assay | Decrease (50 %) | Approved | 29769116 |
DrugRepV_6828 | Dolutegravir | Antiinfectives For Systemic Use | Acquired immunodeficiency syndrome | Human immunodeficiency virus | E92Q/N155H/G163R | | Single-round viral replication assay | Decrease (50 %) | Approved | 29769116 |
DrugRepV_6829 | Cabotegravir | Antiviral | Acquired immunodeficiency syndrome | Human immunodeficiency virus | T66I/T97A/E157Q | | Single-round viral replication assay | Decrease (50 %) | Phase I | 29769116 |
DrugRepV_6830 | Cabotegravir | Antiviral | Acquired immunodeficiency syndrome | Human immunodeficiency virus | T97A/Y143R/N155H | | Single-round viral replication assay | Decrease (50 %) | Phase I | 29769116 |
DrugRepV_6831 | Cabotegravir | Antiviral | Acquired immunodeficiency syndrome | Human immunodeficiency virus | G140S/Y143R/N155H | | Single-round viral replication assay | Decrease (50 %) | Phase I | 29769116 |
DrugRepV_6832 | Cabotegravir | Antiviral | Acquired immunodeficiency syndrome | Human immunodeficiency virus | E92Q/N155H/G163R | | Single-round viral replication assay | Decrease (50 %) | Phase I | 29769116 |
DrugRepV_6833 | Bictegravir | Antiinfectives For Systemic Use | Acquired immunodeficiency syndrome | Human immunodeficiency virus | T66I/T97A/E157Q | | Single-round viral replication assay | Decrease (50 %) | Approved | 29769116 |
DrugRepV_6834 | Bictegravir | Antiinfectives For Systemic Use | Acquired immunodeficiency syndrome | Human immunodeficiency virus | T97A/Y143R/N155H | | Single-round viral replication assay | Decrease (50 %) | Approved | 29769116 |
DrugRepV_6835 | Bictegravir | Antiinfectives For Systemic Use | Acquired immunodeficiency syndrome | Human immunodeficiency virus | G140S/Y143R/N155H | | Single-round viral replication assay | Decrease (50 %) | Approved | 29769116 |
DrugRepV_6836 | Bictegravir | Antiinfectives For Systemic Use | Acquired immunodeficiency syndrome | Human immunodeficiency virus | E92Q/N155H/G163R | | Single-round viral replication assay | Decrease (50 %) | Approved | 29769116 |
DrugRepV_6837 | Raltegravir | Antiinfectives For Systemic Use | Acquired immunodeficiency syndrome | Human immunodeficiency virus | T97A/G140S/Q148H | | Single-round viral replication assay | Decrease (50 %) | Approved | 29769116 |
DrugRepV_6838 | Raltegravir | Antiinfectives For Systemic Use | Acquired immunodeficiency syndrome | Human immunodeficiency virus | E138A/G140S/Q148H | | Single-round viral replication assay | Decrease (50 %) | Approved | 29769116 |
DrugRepV_6839 | Raltegravir | Antiinfectives For Systemic Use | Acquired immunodeficiency syndrome | Human immunodeficiency virus | E138K/G140S/Q148H | | Single-round viral replication assay | Decrease (50 %) | Approved | 29769116 |
DrugRepV_6840 | Raltegravir | Antiinfectives For Systemic Use | Acquired immunodeficiency syndrome | Human immunodeficiency virus | G140S/Y143R/Q148H | | Single-round viral replication assay | Decrease (50 %) | Approved | 29769116 |
DrugRepV_6841 | Raltegravir | Antiinfectives For Systemic Use | Acquired immunodeficiency syndrome | Human immunodeficiency virus | G140S/Q148H/N155H | | Single-round viral replication assay | Decrease (50 %) | Approved | 29769116 |
DrugRepV_6842 | Raltegravir | Antiinfectives For Systemic Use | Acquired immunodeficiency syndrome | Human immunodeficiency virus | G140S/Q148H/G163K | | Single-round viral replication assay | Decrease (50 %) | Approved | 29769116 |
DrugRepV_6843 | Elvitegravir | Antiinfectives For Systemic Use | Acquired immunodeficiency syndrome | Human immunodeficiency virus | T97A/G140S/Q148H | | Single-round viral replication assay | Decrease (50 %) | Approved | 29769116 |
DrugRepV_6844 | Elvitegravir | Antiinfectives For Systemic Use | Acquired immunodeficiency syndrome | Human immunodeficiency virus | E138A/G140S/Q148H | | Single-round viral replication assay | Decrease (50 %) | Approved | 29769116 |
DrugRepV_6845 | Elvitegravir | Antiinfectives For Systemic Use | Acquired immunodeficiency syndrome | Human immunodeficiency virus | E138K/G140S/Q148H | | Single-round viral replication assay | Decrease (50 %) | Approved | 29769116 |
DrugRepV_6846 | Elvitegravir | Antiinfectives For Systemic Use | Acquired immunodeficiency syndrome | Human immunodeficiency virus | G140S/Y143R/Q148H | | Single-round viral replication assay | Decrease (50 %) | Approved | 29769116 |
DrugRepV_6847 | Elvitegravir | Antiinfectives For Systemic Use | Acquired immunodeficiency syndrome | Human immunodeficiency virus | G140S/Q148H/N155H | | Single-round viral replication assay | Decrease (50 %) | Approved | 29769116 |
DrugRepV_6848 | Elvitegravir | Antiinfectives For Systemic Use | Acquired immunodeficiency syndrome | Human immunodeficiency virus | G140S/Q148H/G163K | | Single-round viral replication assay | Decrease (50 %) | Approved | 29769116 |
DrugRepV_6849 | Dolutegravir | Antiinfectives For Systemic Use | Acquired immunodeficiency syndrome | Human immunodeficiency virus | T97A/G140S/Q148H | | Single-round viral replication assay | Decrease (50 %) | Approved | 29769116 |
DrugRepV_6850 | Dolutegravir | Antiinfectives For Systemic Use | Acquired immunodeficiency syndrome | Human immunodeficiency virus | E138A/G140S/Q148H | | Single-round viral replication assay | Decrease (50 %) | Approved | 29769116 |
DrugRepV_6851 | Dolutegravir | Antiinfectives For Systemic Use | Acquired immunodeficiency syndrome | Human immunodeficiency virus | E138K/G140S/Q148H | | Single-round viral replication assay | Decrease (50 %) | Approved | 29769116 |
DrugRepV_6852 | Dolutegravir | Antiinfectives For Systemic Use | Acquired immunodeficiency syndrome | Human immunodeficiency virus | G140S/Y143R/Q148H | | Single-round viral replication assay | Decrease (50 %) | Approved | 29769116 |
DrugRepV_6853 | Dolutegravir | Antiinfectives For Systemic Use | Acquired immunodeficiency syndrome | Human immunodeficiency virus | G140S/Q148H/N155H | | Single-round viral replication assay | Decrease (50 %) | Approved | 29769116 |
DrugRepV_6854 | Dolutegravir | Antiinfectives For Systemic Use | Acquired immunodeficiency syndrome | Human immunodeficiency virus | G140S/Q148H/G163K | | Single-round viral replication assay | Decrease (50 %) | Approved | 29769116 |
DrugRepV_6855 | Cabotegravir | Antiviral | Acquired immunodeficiency syndrome | Human immunodeficiency virus | T97A/G140S/Q148H | | Single-round viral replication assay | Decrease (50 %) | Phase I | 29769116 |
DrugRepV_6856 | Cabotegravir | Antiviral | Acquired immunodeficiency syndrome | Human immunodeficiency virus | E138A/G140S/Q148H | | Single-round viral replication assay | Decrease (50 %) | Phase I | 29769116 |
DrugRepV_6857 | Cabotegravir | Antiviral | Acquired immunodeficiency syndrome | Human immunodeficiency virus | E138K/G140S/Q148H | | Single-round viral replication assay | Decrease (50 %) | Phase I | 29769116 |
DrugRepV_6858 | Cabotegravir | Antiviral | Acquired immunodeficiency syndrome | Human immunodeficiency virus | G140S/Y143R/Q148H | | Single-round viral replication assay | Decrease (50 %) | Phase I | 29769116 |
DrugRepV_6859 | Cabotegravir | Antiviral | Acquired immunodeficiency syndrome | Human immunodeficiency virus | G140S/Q148H/N155H | | Single-round viral replication assay | Decrease (50 %) | Phase I | 29769116 |
DrugRepV_6860 | Cabotegravir | Antiviral | Acquired immunodeficiency syndrome | Human immunodeficiency virus | G140S/Q148H/G163K | | Single-round viral replication assay | Decrease (50 %) | Phase I | 29769116 |
DrugRepV_6861 | Bictegravir | Antiinfectives For Systemic Use | Acquired immunodeficiency syndrome | Human immunodeficiency virus | T97A/G140S/Q148H | | Single-round viral replication assay | Decrease (50 %) | Approved | 29769116 |
DrugRepV_6862 | Bictegravir | Antiinfectives For Systemic Use | Acquired immunodeficiency syndrome | Human immunodeficiency virus | E138A/G140S/Q148H | | Single-round viral replication assay | Decrease (50 %) | Approved | 29769116 |
DrugRepV_6863 | Bictegravir | Antiinfectives For Systemic Use | Acquired immunodeficiency syndrome | Human immunodeficiency virus | E138K/G140S/Q148H | | Single-round viral replication assay | Decrease (50 %) | Approved | 29769116 |
DrugRepV_6864 | Bictegravir | Antiinfectives For Systemic Use | Acquired immunodeficiency syndrome | Human immunodeficiency virus | G140S/Y143R/Q148H | | Single-round viral replication assay | Decrease (50 %) | Approved | 29769116 |
DrugRepV_6865 | Bictegravir | Antiinfectives For Systemic Use | Acquired immunodeficiency syndrome | Human immunodeficiency virus | G140S/Q148H/N155H | | Single-round viral replication assay | Decrease (50 %) | Approved | 29769116 |
DrugRepV_6866 | Bictegravir | Antiinfectives For Systemic Use | Acquired immunodeficiency syndrome | Human immunodeficiency virus | G140S/Q148H/G163K | | Single-round viral replication assay | Decrease (50 %) | Approved | 29769116 |